SCHEMBL4448529

SCHEMBL4448529

Cln1cnc2cnccc21

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FGFR1 P11362 1/20 0.53
LTA4H P09960 1/20 0.38
ALDH1A1 P00352 3/20 0.38
KDM4E B2RXH2 2/20 0.38
MKNK1 Q9BUB5 2/20 0.37
MKNK2 Q9HBH9 2/20 0.37
TGFBR1 P36897 1/20 0.35
JAK2 O60674 1/20 0.35
JAK3 P52333 1/20 0.35
ATM Q13315 1/20 0.35
MET P08581 1/20 0.35
HCAR1 Q9BXC0 1/20 0.33
NPC1 O15118 1/20 0.33
LMNA P02545 1/20 0.33
TP53 P04637 1/20 0.33
MAPT P10636 1/20 0.33
HPGD P15428 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
HSD17B10 Q99714 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL34465814 0.80 FGFR1 (0.42) FGFR1LTA4HALDH1A1KDM4EMKNK1
SCHEMBL4059255 0.75 FGFR1 (0.53) FGFR1LTA4HALDH1A1KDM4EMKNK1
SCHEMBL29593970 0.75 FGFR1 (0.53) FGFR1LTA4HALDH1A1KDM4EMKNK1
SCHEMBL256337 0.75 FGFR1 (0.53) FGFR1LTA4HALDH1A1KDM4EMKNK1
SCHEMBL18330920 0.75 FGFR1 (0.53) FGFR1LTA4HALDH1A1KDM4EMKNK1
SCHEMBL25291568 0.75 FGFR1 (0.53) FGFR1LTA4HALDH1A1KDM4EMKNK1
SCHEMBL5030414 0.72 FGFR1 (0.46) FGFR1LTA4HALDH1A1KDM4EMKNK1
SCHEMBL277760 0.71 TDP1 (0.54) FGFR1LMNAHPGDSMN1; SMN2HSD17B10
SCHEMBL1701476 0.71 FGFR1 (0.49) FGFR1LTA4HALDH1A1KDM4EMKNK1
SCHEMBL1106481 0.71 FGFR1 (0.49) FGFR1LTA4HALDH1A1KDM4EJAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12312353-B2 Piperidinyl-methyl-purineamines as NSD2 inhibitors and anti-cancer agents NOVARTIS AG (CH) 2025-05-27 US disclosed
US-20230002388-A1 PIPERIDINYL-METHYL-PURINEAMINES AS NSD2 INHIBITORS AND ANTI-CANCER AGENTS CHINA NOVARTIS INSTITUTES FOR BIOMEDICAL RESEARCH CO., LTD. (CN) 2023-01-05 US disclosed
US-11420970-B1 Piperidinyl-methyl-purineamines as NSD2 inhibitors and anti-cancer agents NOVARTIS AG (CH) 2022-08-23 US disclosed
US-20090270431-A1 Cyclopentenol Nucleoside Compounds Intermediates for their Synthesis and Methods of Treating Viral Infections THE UNIVERSITY OF GEORGIA RESEARCH FOUNDATION (US) 2009-10-29 US disclosed
WO-2007047793-A2 CYCLOPENTENOL NUCLEOSIDE COMPOUNDS, INTERMEDIATES FOR THEIR SYNTHESIS AND METHODS OF TREATING VIRAL INFECTIONS UNIVERSITY OF GEORGIA RESEARCH FOUNDATION, INC. (US) 2007-04-26 WO disclosed
US-5446139-A Purine analog nucleoside and nucleotide compounds BOEHRINGER MANNHEIM GMBH (DE) 1995-08-29 US disclosed
EP-0038568-B1 SYNTHESIS OF DEAZAPURINE NUCLEOSIDES THE WELLCOME FOUNDATION LIMITED (GB) 1983-07-20 EP disclosed
US-4347315-A FORMING 4-SUBSTITUTED 1-B-D-RIBOFURANOSYL-1H-IMIDAZO(4,5-C)PYRIDINES FROM RIBOSE-1-PHOSPHATE BURROUGHS WELLCOME CO. (US) 1982-08-31 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12312353-B2 Piperidinyl-methyl-purineamines as NSD2 inhibitors and anti-cancer agents NSD2, NSD1, NSD3 FGFR1 4459/4885LTA4H 4414/4885ALDH1A1 3642/4885
US-11420970-B1 Piperidinyl-methyl-purineamines as NSD2 inhibitors and anti-cancer agents NSD2, NSD1, NSD3 FGFR1 4459/4885LTA4H 4414/4885ALDH1A1 3642/4885
US-20090270431-A1 Cyclopentenol Nucleoside Compounds Intermediates for their Synthesis and Methods of Treating Viral Infections REV1, NSUN2, ORC3 FGFR1 2172/4885LTA4H 1759/4885ALDH1A1 1749/4885
US-20230002388-A1 PIPERIDINYL-METHYL-PURINEAMINES AS NSD2 INHIBITORS AND ANTI-CANCER AGENTS NSD2, NSD1, NSD3 FGFR1 4459/4885LTA4H 4414/4885ALDH1A1 3642/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.