SCHEMBL4449227

SCHEMBL4449227

CNc1ccnc(C)c1C

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 1/20 0.37
ROCK1 Q13464 1/20 0.37
CDC42BPA Q5VT25 1/20 0.37
CDC42BPB Q9Y5S2 1/20 0.37
SLC40A1 Q9NP59 1/20 0.36
CYP2A6 P11509 1/20 0.35
NOS3 P29474 1/20 0.33
NOS2 P35228 1/20 0.33
CYP1A2 P05177 2/20 0.33
CYP3A4 P08684 2/20 0.33
CYP2C19 P33261 2/20 0.33
CYP2C9 P11712 1/20 0.33
HSD17B10 Q99714 1/20 0.33
HTR1A P08908 3/20 0.32
ADRA1D P25100 3/20 0.32
ADRA1A P35348 3/20 0.32
ADRA1B P35368 3/20 0.32
AOC1 P19801 2/20 0.31
AOC3 Q16853 2/20 0.31
GRM1 Q13255 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21598449 0.79 CA12 (0.37) CYP2A6NOS3NOS2HTR1AADRA1D
SCHEMBL30147759 0.79 CA12 (0.37) CYP2A6NOS3NOS2HTR1AADRA1D
SCHEMBL17547276 0.77 METAP2 (0.37) ROCK2ROCK1CDC42BPACDC42BPBSLC40A1
SCHEMBL21092874 0.77 ROCK2 (0.35) ROCK2ROCK1CDC42BPACDC42BPBSLC40A1
SCHEMBL23999693 0.77 NOS2 (0.56) ROCK2ROCK1CDC42BPACDC42BPBSLC40A1
SCHEMBL10883659 0.77 ROCK2 (0.35) ROCK2ROCK1CDC42BPACDC42BPBSLC40A1
SCHEMBL27578120 0.74 CYP2A6 (0.31) ROCK1CYP2A6PDE3BPDE3A
SCHEMBL4272874 0.74 ESR2 (0.34) CYP2A6CCR1CCR5CCR8PDE3B
SCHEMBL17667913 0.74 PDE3B (0.35) ROCK2ROCK1CDC42BPACDC42BPBNOS3
SCHEMBL8801086 0.73 PIK3C3 (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7595413-B2 Phosphine-substituted vinyl containing metallocene catalyst, preparation process and the application of the same PETROCHINA COMPANY LIMITED (CN) 2009-09-29 US claimed
WO-2021226517-A1 AKT3 MODULATORS GEORGIAMUNE LLC (US) 2021-11-11 WO disclosed
EP-1958969-A1 A phosphine-substituted vinyl containing metallocene catalyst, preparation process and the application of the same Petrochina Company Limited (CN) 2008-08-20 EP disclosed