SCHEMBL4452402

SCHEMBL4452402

O=C1NC(=O)C2(CC34CN(C(=O)O)CC(=O)N3CC3(CCN(Cc5ccccc5)CC3)N4)C=CC=CC12

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 11/20 0.33
OPRM1 P35372 1/20 0.33
OPRD1 P41143 1/20 0.33
OPRK1 P41145 1/20 0.33
OPRL1 P41146 1/20 0.33
CYP3A4 P08684 6/20 0.33
CHRM2 P08172 3/20 0.33
ALDH1A1 P00352 3/20 0.33
CHRM3 P20309 1/20 0.33
TSHR P16473 4/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
USP2 O75604 2/20 0.32
HSD11B1 P28845 1/20 0.32
MAPK1 P28482 2/20 0.32
MEN1 O00255 1/20 0.32
HTT P42858 1/20 0.32
KMT2A Q03164 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
HRH3 Q9Y5N1 1/20 0.31
CYP2C19 P33261 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4246121 0.80 F10 (0.51) CYP2D6CYP3A4ALDH1A1TSHRUSP2
SCHEMBL4237209 0.79 CYP2D6 (0.41) CYP2D6OPRM1OPRD1OPRK1OPRL1
SCHEMBL4454901 0.79 CYP2D6 (0.42) CYP2D6OPRM1OPRD1OPRK1OPRL1
SCHEMBL4522977 0.77 CYP2D6 (0.47) CYP2D6OPRM1OPRD1OPRK1OPRL1
SCHEMBL4519652 0.75 CYP2D6 (0.41) CYP2D6OPRM1OPRD1OPRK1OPRL1
SCHEMBL4454104 0.70 POLB (0.44) ALDH1A1MAPK1MEN1HTTKMT2A
SCHEMBL6079416 0.69 CYP2D6 (0.45) CYP2D6OPRD1OPRK1CYP3A4CHRM2
SCHEMBL4449570 0.67 POLB (0.43) ALDH1A1L3MBTL1MEN1HTTKMT2A
SCHEMBL12610592 0.66 DRD4 (0.48) CYP2D6CYP3A4
SCHEMBL4526398 0.65 CYP2D6 (0.48) CYP2D6CYP3A4CHRM2ALDH1A1CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2020411-A1 SPIRO TETRACYCLIC COMPOUND MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 2009-02-04 EP disclosed