SCHEMBL4454901

SCHEMBL4454901

CNCC12CN(C(=O)O)CC(=O)N1CC1(CCN(Cc3ccccc3)CC1)N2

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 13/20 0.42
CHRM2 P08172 4/20 0.39
CHRM3 P20309 2/20 0.39
ALDH1A1 P00352 5/20 0.39
MAPK1 P28482 2/20 0.38
CYP3A4 P08684 5/20 0.38
TSHR P16473 4/20 0.38
NPFFR1 Q9GZQ6 1/20 0.37
NPFFR2 Q9Y5X5 1/20 0.37
OPRM1 P35372 1/20 0.37
OPRD1 P41143 1/20 0.37
OPRK1 P41145 1/20 0.37
OPRL1 P41146 1/20 0.37
USP2 O75604 1/20 0.37
KDM4E B2RXH2 1/20 0.37
CYP2C19 P33261 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4237209 0.87 CYP2D6 (0.41) CYP2D6CHRM2CHRM3ALDH1A1MAPK1
SCHEMBL4522977 0.86 CYP2D6 (0.47) CYP2D6CHRM2CHRM3ALDH1A1MAPK1
SCHEMBL4519652 0.84 CYP2D6 (0.41) CYP2D6CHRM2CHRM3ALDH1A1MAPK1
SCHEMBL4454104 0.80 POLB (0.44) ALDH1A1MAPK1KDM4E
SCHEMBL5322750 0.79 CYP2D6 (0.38) CYP2D6CHRM2CHRM3ALDH1A1CYP3A4
SCHEMBL4452402 0.79 CYP2D6 (0.33) CYP2D6CHRM2CHRM3ALDH1A1MAPK1
SCHEMBL6079416 0.78 CYP2D6 (0.45) CYP2D6CHRM2CHRM3ALDH1A1MAPK1
SCHEMBL4532180 0.77 SIGMAR1 (0.42) CYP2D6CHRM2CHRM3ALDH1A1CYP3A4
SCHEMBL4519880 0.77 CYP2D6 (0.42) CYP2D6CHRM2CHRM3ALDH1A1MAPK1
SCHEMBL4449570 0.76 POLB (0.43) ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2020411-A1 SPIRO TETRACYCLIC COMPOUND MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 2009-02-04 EP disclosed