SCHEMBL4455598

SCHEMBL4455598

C[C@H](NC1CC(=O)OC1OCc1ccccc1)C(=O)NC(=O)c1c[nH]c(CCc2ccc(CC(F)(F)F)cc2)n1

nearest known ligand 0.34

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 5/20 0.34
CASP1 P29466 4/20 0.32
CASP3 P42574 4/20 0.32
CASP7 P55210 4/20 0.32
CASP6 P55212 4/20 0.32
CASP8 Q14790 4/20 0.32
HSD17B2 P37059 1/20 0.31
MMP2 P08253 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL949088 0.93 CASP1 (0.35) CASP1CASP3CASP7CASP6CASP8
SCHEMBL952741 0.93 PDE2A (0.37) PDE2AMMP2
SCHEMBL949112 0.86 CASP1 (0.35) PDE2ACASP1CASP3CASP7CASP6
SCHEMBL952739 0.82 PDE2A (0.40) PDE2ACASP1CASP3CASP7CASP6
SCHEMBL949086 0.81 CASP3 (0.39) CASP1CASP3CASP7CASP6CASP8
SCHEMBL950252 0.81 CASP1 (0.35) CASP1CASP3CASP7CASP6CASP8
SCHEMBL949260 0.78 NAAA (0.34) CASP1CASP3CASP7CASP6CASP8
SCHEMBL948261 0.76 CASP3 (0.35) CASP1CASP3CASP7CASP6CASP8
SCHEMBL948808 0.75 CASP3 (0.38) CASP1CASP3CASP7CASP6CASP8
SCHEMBL949530 0.74 CASP3 (0.38) CASP1CASP3CASP7CASP6CASP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2123665-A2 Inhibitors of interleukin-1Beta converting enzyme Vertex Pharmaceuticals Incorporated (US) 2009-11-25 EP disclosed