Bromide

Bromide

SCHEMBL4455959

Br.c1ccc(CCc2cc(-c3ccccc3)nc3ccccc23)cc1

nearest known ligand 0.53

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ACHE known ✓ P22303 1/20 0.53
TACR3 P29371 2/20 0.50
LMNA P02545 2/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
KDM4E B2RXH2 2/20 0.49
PDE10A Q9Y233 1/20 0.49
HPGD P15428 1/20 0.49
ACP1 P24666 2/20 0.47
SLC2A1 P11166 1/20 0.47
DHODH Q02127 2/20 0.46
CYP2C9 P11712 1/20 0.46
ACACA Q13085 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28619856 0.83 ACHE (0.56) ACHETACR3LMNASMN1; SMN2KDM4E
SCHEMBL1259674 0.79 ACHE (0.59) ACHETACR3LMNASMN1; SMN2KDM4E
SCHEMBL27917367 0.79 DHODH (0.58) ACHETACR3LMNASMN1; SMN2HPGD
SCHEMBL27367367 0.79 ACHE (0.51) ACHETACR3LMNASMN1; SMN2KDM4E
SCHEMBL11172886 0.78 KDM4E (0.55) ACHELMNASMN1; SMN2KDM4EPDE10A
SCHEMBL10671292 0.78 PDE10A (0.58) ACHETACR3LMNASMN1; SMN2KDM4E
SCHEMBL20809331 0.78 ACHE (0.50) ACHETACR3LMNASMN1; SMN2KDM4E
SCHEMBL8675109 0.78 ACHE (0.50) ACHETACR3LMNASMN1; SMN2KDM4E
SCHEMBL9988793 0.78 DHODH (0.53) ACHETACR3LMNASMN1; SMN2KDM4E
SCHEMBL8091105 0.78 ACHE (0.54) ACHELMNASMN1; SMN2KDM4EPDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7598390-B2 Fluorescent chemical compounds having high selectivity for double stranded DNA, and methods for their use Life Technologies Corporation (US) 2009-10-06 US disclosed
US-20060263844-A1 Flourescent chemical compounds having high selectivity for double standard DNA, and methods for their use MOLECULAR PROBES, INC. 2006-11-23 US disclosed