SCHEMBL4457103

SCHEMBL4457103

NC1=NC(N)(CCc2cccs2)NC=C1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.42
TSHR P16473 2/20 0.39
ADRA2A P08913 3/20 0.36
ADRA2B P18089 3/20 0.36
ADRA2C P18825 3/20 0.36
L3MBTL1 Q9Y468 2/20 0.33
ALDH1A1 P00352 1/20 0.33
POLB P06746 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
GPR84 Q9NQS5 1/20 0.33
ADRA1D P25100 2/20 0.32
HSD17B10 Q99714 1/20 0.32
HPGD P15428 1/20 0.32
PIK3CD O00329 1/20 0.32
PIK3CB P42338 1/20 0.32
HCAR3 P49019 1/20 0.32
TDP1 Q9NUW8 1/20 0.31
PTGS1 P23219 1/20 0.31
PTGS2 P35354 1/20 0.31
MGMT P16455 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4455633 0.70 DRD2 (0.40) L3MBTL1ALDH1A1SMN1; SMN2HSD17B10HPGD
SCHEMBL2069431 0.65 SLC6A3 (0.33) ALDH1A1TDP1
SCHEMBL2069292 0.65 SLC6A2 (0.32)
SCHEMBL2030841 0.64 TAAR1 (0.71) TAAR1TSHRADRA2AADRA2BADRA2C
SCHEMBL31617182 0.62 TAAR1 (0.35) TAAR1TSHRADRA2AADRA2BADRA2C
SCHEMBL244450 0.61
SCHEMBL72881 0.61
SCHEMBL20146704 0.61 TAAR1 (0.73) TAAR1TSHRADRA2AADRA2BADRA2C
SCHEMBL20135772 0.61 TAAR1 (0.73) TAAR1TSHRADRA2AADRA2BADRA2C
SCHEMBL121154 0.61

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009017838-A2 COMBINATIONS OF JAK-2 INHIBITORS AND OTHER AGENTS EXELIXIS, INC. (US) 2009-02-05 WO claimed