SCHEMBL4458353

SCHEMBL4458353

NC1=NC(N)(Cc2cc(-c3cnccn3)no2)NC=C1

nearest known ligand 0.35

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
IGF1R P08069 1/20 0.35
CYP2E1 P05181 1/20 0.32
CYP2A6 P11509 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2B6 P20813 1/20 0.32
CYP2C19 P33261 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4464611 0.73 SMN1; SMN2 (0.47) IGF1RCYP2C9
SCHEMBL4459263 0.65 CHRNA7 (0.40) CYP2A6CYP2C9
SCHEMBL4472365 0.64 DHFR (0.39)
SCHEMBL28854929 0.60 CYP2C9 (0.36) IGF1RCYP2E1CYP2A6CYP2C9CYP2B6
SCHEMBL29454745 0.57 NISCH (0.50) CYP2C9CYP2C19
SCHEMBL78566 0.57 NISCH (0.50) CYP2C9CYP2C19
SCHEMBL29598957 0.57 NISCH (0.50) CYP2C9CYP2C19
SCHEMBL27790030 0.57 NPC1 (0.35) CYP2E1CYP2A6CYP2C9CYP2B6CYP2C19
SCHEMBL11836404 0.57 IGF1R (0.40) IGF1R
SCHEMBL4466158 0.56 VHL (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009017838-A2 COMBINATIONS OF JAK-2 INHIBITORS AND OTHER AGENTS EXELIXIS, INC. (US) 2009-02-05 WO disclosed