SCHEMBL4458987

SCHEMBL4458987

Fc1ccccc1C(F)(F)N(F)F.NCc1ccc(F)cc1F

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 4/20 0.38
AGXT P21549 2/20 0.38
KCNN4 O15554 4/20 0.33
HTR2A P28223 3/20 0.33
HTR2C P28335 3/20 0.33
MAPK14 Q16539 1/20 0.33
RIPK1 Q13546 2/20 0.32
CHRM5 P08912 1/20 0.32
KCNE1 P15382 1/20 0.32
KCNQ1 P51787 1/20 0.32
KDM4E B2RXH2 2/20 0.32
MPO P05164 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
NFE2L2 Q16236 1/20 0.32
TAAR1 Q96RJ0 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL554230 0.78 KCNN4 (0.37) KCNN4KCNE1KCNQ1NFE2L2
SCHEMBL113852 0.76 IDO1 (0.59) IDO1AGXTHTR2AHTR2CKDM4E
SCHEMBL26625794 0.76 IDO1 (0.59) IDO1AGXTHTR2AHTR2CKDM4E
Trifluoroacetic Acid SCHEMBL4243585 0.69 IDO1 (0.44) IDO1AGXTKCNN4HTR2AHTR2C
SCHEMBL8356956 0.67 IDO1 (0.42) IDO1AGXTKDM4EMPOSMN1; SMN2
SCHEMBL4458984 0.66 IDO1 (0.48) IDO1AGXTHTR2AHTR2CMAPK14
SCHEMBL109671 0.66 IDO1 (0.65) IDO1AGXTMPO
SCHEMBL888536 0.64 KCNN4 (0.33) KCNN4KCNE1KCNQ1
SCHEMBL18783726 0.64 MAPK14 (0.56) IDO1AGXTMAPK14KDM4E
SCHEMBL11623483 0.64 IDO1 (0.41) IDO1KCNN4MPOTAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0819000-B1 NODULISPORIC ACID DERIVATIVES MERCK & CO INC (US) 2009-07-08 EP disclosed