SCHEMBL4458992

SCHEMBL4458992

COc1c(C(C)(C)C)cc(-c2cccc(C3CCN(C(=O)O)C(C(C)(C)C)C3)n2)cc1C(C)(C)C

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
FFAR4 Q5NUL3 5/20 0.35
ADORA2A P29274 1/20 0.35
ADORA1 P30542 1/20 0.35
UBE2M P61081 3/20 0.34
DCUN1D1 Q96GG9 3/20 0.34
TNFRSF1A P19438 1/20 0.33
HTR1A P08908 3/20 0.32
DRD2 P14416 3/20 0.32
DRD4 P21917 3/20 0.32
KCNH2 Q12809 2/20 0.32
HDAC8 Q9BY41 2/20 0.32
FPR2 P25090 1/20 0.32
ROCK2 O75116 1/20 0.31
CNR2 P34972 1/20 0.31
ALDH1A1 P00352 1/20 0.30
HTT P42858 1/20 0.30
TAAR1 Q96RJ0 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4456610 0.85 FFAR4 (0.40) FFAR4HTR1ADRD2DRD4KCNH2
SCHEMBL4451812 0.82 FFAR4 (0.41) FFAR4HTR1ADRD2DRD4KCNH2
SCHEMBL4462828 0.79 ADORA2A (0.36) FFAR4ADORA2AADORA1TNFRSF1AHTR1A
SCHEMBL4458994 0.78 HTT (0.48) ALDH1A1HTT
SCHEMBL29053049 0.77 DRD4 (0.37) HTR1ADRD2DRD4KCNH2CNR2
Trifluoroacetic Acid SCHEMBL4454113 0.74 PKM (0.39) FFAR4ADORA2AADORA1TNFRSF1AHDAC8
SCHEMBL13959332 0.73 PIM1 (0.41) ADORA2AADORA1FPR2
SCHEMBL4463529 0.71 CXCR3 (0.42) HTR1ADRD2DRD4KCNH2ALDH1A1
SCHEMBL4454107 0.71 IRAK4 (0.39) FFAR4UBE2MDCUN1D1HTR1ADRD2
SCHEMBL13972997 0.71 GRM5 (0.39) ADORA2AADORA1HTR1ADRD2DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090030012-A1 Pyridine, Pyrimidine and Pyrazine Derivatives as Cxcr3 Receptor Modulators MERCK SHARP & DOHME CORP. 2009-01-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090030012-A1 Pyridine, Pyrimidine and Pyrazine Derivatives as Cxcr3 Receptor Modulators CXCR3, CXCR1, CXCR5 FFAR4 212/4885ADORA2A 42/4885ADORA1 67/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.