SCHEMBL4459491

SCHEMBL4459491

NC1=NC=CC(N)(c2ccc(CCN3CCCC3)cc2)N1

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 10/20 0.44
L3MBTL1 Q9Y468 3/20 0.44
MBTD1 Q05BQ5 2/20 0.44
L3MBTL3 Q96JM7 2/20 0.44
TDP1 Q9NUW8 1/20 0.43
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
SLC6A3 Q01959 1/20 0.42
SIGMAR1 Q99720 4/20 0.41
KCNJ1 P48048 1/20 0.36
KCNH2 Q12809 1/20 0.36
TP53BP1 Q12888 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4459064 0.99 HRH3 (0.47) HRH3L3MBTL1MBTD1L3MBTL3TDP1
SCHEMBL4459484 0.73 SLC6A3 (0.44) HRH3L3MBTL1MBTD1L3MBTL3TDP1
SCHEMBL4459061 0.72 HRH3 (0.46) HRH3L3MBTL1MBTD1L3MBTL3TDP1
SCHEMBL4281846 0.71 DRD2 (0.33)
SCHEMBL2911025 0.69 MAPT (0.40) CYP1A2SLC6A3
SCHEMBL4462970 0.69 HRH3 (0.44) HRH3L3MBTL1MBTD1L3MBTL3TDP1
SCHEMBL1877934 0.69 HRH3 (0.68) HRH3L3MBTL1MBTD1L3MBTL3TDP1
SCHEMBL2762024 0.67 HRH3 (0.71) HRH3L3MBTL1MBTD1L3MBTL3TDP1
SCHEMBL2761916 0.67 HRH3 (0.71) HRH3L3MBTL1MBTD1L3MBTL3TDP1
Hydrochloric Acid SCHEMBL916318 0.66 HRH3 (0.69) HRH3L3MBTL1MBTD1L3MBTL3TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009017838-A2 COMBINATIONS OF JAK-2 INHIBITORS AND OTHER AGENTS EXELIXIS, INC. (US) 2009-02-05 WO claimed
WO-2009017838-A2 COMBINATIONS OF JAK-2 INHIBITORS AND OTHER AGENTS EXELIXIS, INC. (US) 2009-02-05 WO disclosed