SCHEMBL4461053

SCHEMBL4461053

NC(=O)CN1CCCC1c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 3/20 0.50
RIPK1 Q13546 2/20 0.50
KDM4E B2RXH2 1/20 0.50
MEN1 O00255 1/20 0.50
ALDH1A1 P00352 1/20 0.50
HPGD P15428 1/20 0.50
KMT2A Q03164 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
CHRNB2 P17787 1/20 0.49
CHRNB4 P30926 1/20 0.49
CHRNA3 P32297 1/20 0.49
CHRNA7 P36544 1/20 0.49
CHRNA4 P43681 1/20 0.49
OPRM1 P35372 2/20 0.48
OPRK1 P41145 2/20 0.48
SIGMAR1 Q99720 1/20 0.47
EPHX2 P34913 2/20 0.45
SCN9A Q15858 1/20 0.44
HSP90AA1 P07900 1/20 0.44
HSP90AB1 P08238 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7493746 0.95 KDM4E (0.55) TACR1RIPK1KDM4EMEN1ALDH1A1
SCHEMBL6092369 0.82 KDM4E (0.58) TACR1RIPK1KDM4EMEN1ALDH1A1
SCHEMBL28945745 0.82 KDM4E (0.58) TACR1RIPK1KDM4EMEN1ALDH1A1
SCHEMBL8227508 0.81 ALDH1A1 (0.48) TACR1RIPK1KDM4EMEN1ALDH1A1
Hydrochloric Acid SCHEMBL12480511 0.81 KDM4E (0.56) TACR1RIPK1KDM4EMEN1ALDH1A1
SCHEMBL10775133 0.81 KDM4E (0.56) TACR1RIPK1KDM4EMEN1ALDH1A1
SCHEMBL10775129 0.81 KDM4E (0.56) TACR1RIPK1KDM4EMEN1ALDH1A1
SCHEMBL4955342 0.80 CHRNB2 (0.55) RIPK1KDM4EMEN1ALDH1A1HPGD
Benzene SCHEMBL11161088 0.80 CHRNB2 (0.55) RIPK1KDM4EMEN1ALDH1A1HPGD
SCHEMBL27512084 0.80 CHRNB2 (0.55) RIPK1KDM4EMEN1ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009017838-A2 COMBINATIONS OF JAK-2 INHIBITORS AND OTHER AGENTS EXELIXIS, INC. (US) 2009-02-05 WO claimed