SCHEMBL4461468

SCHEMBL4461468

Nc1nc(N)c(Cc2cc(-c3ccccc3)no2)c(OCCN2CCCCC2)n1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 4/20 0.47
HRH3 Q9Y5N1 3/20 0.45
IGF1R P08069 2/20 0.44
ADORA2A P29274 2/20 0.43
ADORA1 P30542 2/20 0.43
CXCR1 P25024 1/20 0.42
BACE1 P56817 1/20 0.41
DRD2 P14416 2/20 0.40
DRD4 P21917 2/20 0.40
DRD3 P35462 2/20 0.40
ACP1 P24666 1/20 0.40
ACHE P22303 1/20 0.40
MAOB P27338 1/20 0.40
F2R P25116 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4471578 0.81 IGF1R (0.41) HRH3IGF1R
SCHEMBL4457348 0.80 HRH3 (0.35) HRH3IGF1R
SCHEMBL1787674 0.78 NOTUM (0.58) ADORA2AADORA1
SCHEMBL4459206 0.69 PTPN1 (0.44) PTPN1IGF1RCXCR1BACE1DRD2
SCHEMBL21121935 0.69 CXCR1 (0.79) PTPN1HRH3CXCR1
SCHEMBL21121342 0.69 CXCR1 (0.79) PTPN1HRH3CXCR1
SCHEMBL1789897 0.69 IGF1R (0.59) IGF1R
SCHEMBL4459340 0.68 PTPN1 (0.43) PTPN1IGF1RCXCR1DRD2DRD4
SCHEMBL4907342 0.68 ADORA2A (0.56) ADORA2AADORA1DRD4ACHEMAOB
SCHEMBL1791868 0.67 NOTUM (0.52)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009017838-A2 COMBINATIONS OF JAK-2 INHIBITORS AND OTHER AGENTS EXELIXIS, INC. (US) 2009-02-05 WO claimed