SCHEMBL4462269

SCHEMBL4462269

CC(C)(C)[Si](C)(C)OCC1C(O)C(c2ccccc2)CN1C(=O)O

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 5/20 0.36
SLC6A2 P23975 2/20 0.34
SLC6A4 P31645 2/20 0.34
SLC6A3 Q01959 2/20 0.34
TOP2A P11388 1/20 0.34
TACR1 P25103 2/20 0.34
HTT P42858 1/20 0.33
RORC P51449 1/20 0.33
CHRM2 P08172 1/20 0.32
CHRM4 P08173 1/20 0.32
CHRM5 P08912 1/20 0.32
CHRM1 P11229 1/20 0.32
CHRM3 P20309 1/20 0.32
HRH3 Q9Y5N1 1/20 0.32
KDM1A O60341 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4458157 0.90 TACR1 (0.36) SLC6A4SLC6A3TACR1
SCHEMBL4462143 0.84 RIPK1 (0.36) RIPK1TOP2ATACR1
SCHEMBL21874133 0.77 FKBP1A (0.31)
SCHEMBL4093859 0.76 CCR5 (0.39) RORC
SCHEMBL4111698 0.76 CCR5 (0.39) RORC
SCHEMBL4459909 0.74 TACR1 (0.34) SLC6A4SLC6A3TACR1
SCHEMBL15951884 0.74 RIPK1 (0.36) RIPK1HRH3KDM1A
SCHEMBL4099369 0.74 GRIN2B (0.36) KDM1A
SCHEMBL31703176 0.72
SCHEMBL3619614 0.72

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090042854-A1 Hexahydro-3H-Pyrrolizin-3-Ones Useful as Tachykinin Receptor Antagonists MERCK SHARP & DOHME CORP. 2009-02-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090042854-A1 Hexahydro-3H-Pyrrolizin-3-Ones Useful as Tachykinin Receptor Antagonists TACR1, PROKR1, TACR2 RIPK1 1611/4885SLC6A2 1460/4885SLC6A4 835/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.