SCHEMBL4462415

SCHEMBL4462415

O=C(N[C@H](Cc1ccc(Br)cc1)C(=O)O)c1ccco1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSL P07711 1/20 0.57
FPR2 P25090 2/20 0.56
ALDH1A1 P00352 3/20 0.54
SMN1; SMN2 Q16637 2/20 0.54
NPC1 O15118 1/20 0.54
RAB9A P51151 1/20 0.54
CYP1A2 P05177 1/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2D6 P10635 1/20 0.53
CYP2C9 P11712 1/20 0.53
CYP2C19 P33261 1/20 0.53
TSHR P16473 2/20 0.52
PTPN1 P18031 2/20 0.50
L3MBTL1 Q9Y468 1/20 0.49
KDM4E B2RXH2 1/20 0.48
HSD17B10 Q99714 1/20 0.48
KMT2A Q03164 3/20 0.48
MMP2 P08253 2/20 0.47
MMP1 P03956 1/20 0.47
MMP3 P08254 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4460359 1.00 CTSL (0.57) CTSLFPR2ALDH1A1SMN1; SMN2NPC1
SCHEMBL4461672 1.00 CTSL (0.57) CTSLFPR2ALDH1A1SMN1; SMN2NPC1
SCHEMBL4264475 0.90 CTSL (0.67) CTSLALDH1A1SMN1; SMN2CYP1A2CYP3A4
SCHEMBL4264477 0.90 CTSL (0.67) CTSLALDH1A1SMN1; SMN2CYP1A2CYP3A4
SCHEMBL4267852 0.90 CTSL (0.67) CTSLALDH1A1SMN1; SMN2CYP1A2CYP3A4
SCHEMBL12016785 0.88 CTSL (0.58) CTSLALDH1A1SMN1; SMN2CYP1A2CYP3A4
SCHEMBL4466486 0.86 ALDH1A1 (0.59) CTSLALDH1A1SMN1; SMN2CYP1A2CYP3A4
SCHEMBL4474731 0.86 ALDH1A1 (0.59) CTSLALDH1A1SMN1; SMN2CYP1A2CYP3A4
SCHEMBL4466483 0.86 ALDH1A1 (0.59) CTSLALDH1A1SMN1; SMN2CYP1A2CYP3A4
SCHEMBL838462 0.84 CTSL (0.52) CTSLALDH1A1SMN1; SMN2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090042260-A1 PROCESS FOR PREPARING OPTICALLY ACTIVE (S OR R)-ALPHA-AMINO ACID AND OPTICALLY ACTIVE (R OR S)-ALPHA-AMINO ACID ESTER UBE INDUSTRIES, LTD. (JP) 2009-02-12 US disclosed
EP-1942193-A1 PROCESS FOR PRODUCTION OF OPTICALLY ACTIVE (S OR R)-a-AMINO ACID OR OPTICALLY ACTIVE (S OR R)-a -AMINO ACID ESTER Ube Industries, Ltd. (JP) 2008-07-09 EP disclosed