SCHEMBL44641

SCHEMBL44641

O=S(=O)(N1CCSCC1)N1CCSCC1

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.48
TSHR P16473 4/20 0.46
KMT2A Q03164 2/20 0.46
CA12 O43570 1/20 0.46
CA7 P43166 1/20 0.46
CA14 Q9ULX7 1/20 0.46
KDM4E B2RXH2 1/20 0.44
L3MBTL1 Q9Y468 2/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
LMNA P02545 2/20 0.38
ALDH1A1 P00352 2/20 0.34
MEN1 O00255 1/20 0.34
FDPS P14324 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL1131672 0.97 POLB (0.46) POLBTSHRKMT2ACA12CA7
SCHEMBL9028142 0.89 POLB (0.67) POLBTSHRKMT2ACA12CA7
SCHEMBL11412844 0.79 L3MBTL1 (0.38) TSHRL3MBTL1SMN1; SMN2LMNAALDH1A1
SCHEMBL4067499 0.77 L3MBTL1 (0.41) KMT2AL3MBTL1SMN1; SMN2LMNAALDH1A1
SCHEMBL10751242 0.75
SCHEMBL12303022 0.75 L3MBTL1 (0.40) POLBTSHRKDM4EL3MBTL1SMN1; SMN2
SCHEMBL15693600 0.75 L3MBTL1 (0.36) TSHRL3MBTL1SMN1; SMN2LMNAALDH1A1
SCHEMBL12251556 0.71 LMNA (0.40) TSHRL3MBTL1SMN1; SMN2LMNAALDH1A1
SCHEMBL7697563 0.71 L3MBTL1 (0.34) L3MBTL1LMNA
SCHEMBL13902802 0.71 GAA (0.60) KMT2AKDM4EL3MBTL1SMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 5502 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250129085-A1 SUBSTITUTED IMIDAZO[1,2-B]PYRIDAZINES AS PROTEIN KINASE INHIBITORS SUMITOMO PHARMA AMERICA INC (US) 2025-04-24 US claimed
CN-108699052-B Anthelmintic depsipeptide compounds 勃林格殷格翰动物保健美国公司 2022-04-29 CN claimed
CN-111601593-A P38 kinase inhibitor reduces DUX4 and downstream gene expression for treatment of FSHD 弗尔康医疗公司 2020-08-28 CN claimed
EP-3691620-A1 P38 KINASE INHIBITORS REDUCE DUX4 AND DOWNSTREAM GENE EXPRESSION FOR THE TREATMENT OF FSHD Fulcrum Therapeutics, Inc. (US) 2020-08-12 EP claimed
US-20200061074-A1 METHOD OF TREATMENT THE UNIVERSITY OF MELBOURNE (AU) 2020-02-27 US claimed
WO-2019071147-A1 P38 KINASE INHIBITORS REDUCE DUX4 AND DOWNSTREAM GENE EXPRESSION FOR THE TREATMENT OF FSHD Fulcrum Therapeutics, Inc. (US) 2019-04-11 WO claimed
WO-2018148797-A1 A METHOD OF TREATMENT THE UNIVERSITY OF MELBOURNE (AU) 2018-08-23 WO claimed
US-9695175-B2 Highly selective c-Met inhibitors as anticancer agents CB THERAPEUTICS INC. (KY) 2017-07-04 US claimed
EP-3022198-A1 NOVEL 5-SUBSTITUTED BENZIMIDAZOLIUM COMPOUNDS Boehringer Ingelheim International GmbH (DE) 2016-05-25 EP claimed
EP-1685119-B1 N-ACYLSULFONAMIDE APOPTOSIS PROMOTERS ABBVIE BAHAMAS LTD (BS) 2016-03-09 EP claimed
CN-1296486-A Glucocorticoid-selective anti-inflammatory agents ABBOTT LAB (US) 2001-05-23 CN claimed
WO-2001016128-A1 DIBENZOPYRANS AS GLUCOCORTICOID RECEPTOR ANTAGONISTS FOR TREATMENT OF DIABETES ABBOTT LABORATORIES (US) 2001-03-08 WO claimed
WO-2001004115-A2 NOVEL PROCESS FOR SYNTHESIS OF HETEROARYL-SUBSTITUTED UREA COMPOUNDS BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2001-01-18 WO claimed
EP-1068187-A1 PYRAZOLE INHIBITORS OF CYTOKINE PRODUCTION ABBOTT LABORATORIES (US) 2001-01-17 EP claimed
EP-1053240-A1 GLUCOCORTICOID-SELECTIVE ANTIINFLAMMATORY AGENTS Abbott Laboratories (US) 2000-11-22 EP claimed
EP-0986384-A1 INHIBITORS OF PROTEIN ISOPRENYL TRANSFERASES UNIVERSITY OF PITTSBURGH (US) 2000-03-22 EP claimed
WO-1999051580-A1 PYRAZOLE INHIBITORS OF CYTOKINE PRODUCTION ABBOTT LABORATORIES (US) 1999-10-14 WO claimed
WO-1999041257-A1 GLUCOCORTICOID-SELECTIVE ANTIINFLAMMATORY AGENTS ABBOTT LABORATORIES (US) 1999-08-19 WO claimed
WO-1998050030-A1 INHIBITORS OF PROTEIN ISOPRENYL TRANSFERASES UNIVERSITY OF PITTSBURGH (US) 1998-11-12 WO claimed
WO-1995029689-A1 N-CARBOXYALKYL DERIVATIVES AS ANTIDEGENERATIVE ACTIVE AGENTS MERCK & CO., INC. (US) 1995-11-09 WO claimed