SCHEMBL4464235

SCHEMBL4464235

O=C(NS(=O)(=O)c1ccc(Br)cc1)c1ccccc1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 7/20 0.71
PTGS1 P23219 5/20 0.71
FLT1 P17948 3/20 0.71
FLT4 P35916 3/20 0.71
KDR P35968 3/20 0.71
MEN1 O00255 1/20 0.71
LMNA P02545 1/20 0.71
KMT2A Q03164 1/20 0.71
L3MBTL1 Q9Y468 1/20 0.71
EGFR P00533 4/20 0.61
BLM P54132 1/20 0.57
ERBB2 P04626 1/20 0.56
CA1 P00915 1/20 0.56
CA2 P00918 1/20 0.56
MMP1 P03956 1/20 0.56
MMP2 P08253 1/20 0.56
MMP9 P14780 1/20 0.56
MMP8 P22894 1/20 0.56
MMP13 P45452 1/20 0.56
BCL2L1 Q07817 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24347999 0.93 PTGS2 (0.67) PTGS2PTGS1FLT1FLT4KDR
SCHEMBL174010 0.87 FLT1 (0.77) PTGS2PTGS1FLT1FLT4KDR
Potassium SCHEMBL30358590 0.85 FLT1 (0.74) PTGS2PTGS1FLT1FLT4KDR
SCHEMBL29011132 0.85 FLT1 (0.74) PTGS2PTGS1FLT1FLT4KDR
SCHEMBL8424044 0.84 FLT1 (0.73) PTGS2PTGS1FLT1FLT4KDR
SCHEMBL5931288 0.83 FLT1 (0.71) PTGS2PTGS1FLT1FLT4KDR
SCHEMBL7367486 0.83 PTGS2 (0.68) PTGS2PTGS1FLT1FLT4KDR
SCHEMBL5931087 0.83 PTGS2 (0.71) PTGS2PTGS1FLT1FLT4KDR
Sulfabenzamide SCHEMBL93841 0.83 KMT2A (1.00) PTGS2PTGS1FLT1FLT4KDR
SCHEMBL28698398 0.83 PTGS2 (0.71) PTGS2PTGS1FLT1FLT4KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114059090-B Preparation method of benzo [ e ] [1,4,3] oxathiazine-1, 1-dioxide derivative 福州大学 2023-11-21 CN disclosed
CN-114059090-A Preparation method of benzo [ e ] [1,4,3] oxathiazine-1, 1-dioxide derivative 福州大学 2022-02-18 CN disclosed
US-7629366-B2 Aminoalcohol derivatives FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2009-12-08 US disclosed
US-7446222-B2 Phenyl compounds GLAXO GROUP LIMITED (GB) 2008-11-04 US disclosed
US-20060235057-A1 Phenyl compounds GLAXO GROUP LIMITED (GB) 2006-10-19 US disclosed
CN-1802355-A Aminoalcohol derivatives FUJISAWA PHARMACEUTICAL CO (JP) 2006-07-12 CN disclosed
US-20060100252-A1 Aminoalcohol derivatives FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2006-05-11 US disclosed
US-7037938-B2 Aminoalcohol derivatives ASTELLAS PHARMA INC. (JP) 2006-05-02 US disclosed
EP-1556330-A2 PHENYL COMPOUNDS GLAXO GROUP LIMITED (GB) 2005-07-27 EP disclosed
EP-1546086-A2 AMINOALCOHOL DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2005-06-29 EP disclosed
WO-2004039753-A2 PHENYL COMPOUNDS GLAXO GROUP LIMITED (GB) 2004-05-13 WO disclosed
US-20040006143-A1 For therapy of urinary incontinence FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-01-08 US disclosed
WO-2004002939-A2 AMINOALCOHOL DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-01-08 WO disclosed
EP-0189305-A2 Peptide derivatives ICI AMERICAS INC. (US) 1986-07-30 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060235057-A1 Phenyl compounds RXRB, CYP2C9, RXFP1 PTGS2 2262/4885PTGS1 1686/4885FLT1 1427/4885
US-20060100252-A1 Aminoalcohol derivatives H1-0, CHRM2, CHRM1 PTGS2 3088/4885PTGS1 2713/4885FLT1 4151/4885
US-20040006143-A1 For therapy of urinary incontinence H1-0, HRH2, H1-2 PTGS2 1311/4885PTGS1 1072/4885FLT1 4557/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.