SCHEMBL4465210

SCHEMBL4465210

O=C(NCCc1ccccc1Cl)c1cc(-c2c[nH]c(=O)cn2)ccc1Cl

nearest known ligand 0.72

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 13/20 0.72
ABCB11 O95342 1/20 0.57
HIF1A Q16665 2/20 0.51
POLB P06746 2/20 0.47
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
KDM4E B2RXH2 1/20 0.46
MEN1 O00255 1/20 0.46
ALDH1A1 P00352 1/20 0.46
GAA P10253 1/20 0.46
MAPT P10636 1/20 0.46
HPGD P15428 1/20 0.46
KMT2A Q03164 1/20 0.46
ROCK2 O75116 1/20 0.43
ROCK1 Q13464 1/20 0.43
TP53 P04637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2169310 0.82 P2RX7 (0.67) P2RX7ABCB11HIF1APOLBNPC1
SCHEMBL2168393 0.82 P2RX7 (1.00) P2RX7ABCB11HIF1AKMT2A
SCHEMBL4465535 0.82 P2RX7 (0.69) P2RX7ABCB11HIF1AROCK2ROCK1
SCHEMBL4471577 0.80 P2RX7 (0.69) P2RX7ABCB11HIF1APOLBNPC1
SCHEMBL4472433 0.77 P2RX7 (0.72) P2RX7ABCB11HIF1APOLBKDM4E
SCHEMBL5118090 0.76 P2RX7 (0.67) P2RX7ABCB11HIF1APOLBNPC1
SCHEMBL4482089 0.75 P2RX7 (1.00) P2RX7ABCB11HIF1AROCK2ROCK1
SCHEMBL14609832 0.74 P2RX7 (0.71) P2RX7ABCB11HIF1APOLBKDM4E
SCHEMBL4470885 0.74 P2RX7 (0.62) P2RX7ABCB11HIF1ATP53
SCHEMBL5111555 0.74 P2RX7 (0.66) P2RX7ABCB11HIF1APOLBNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7553972-B2 Benzamide inhibitors of the P2X7 receptor PFIZER, INC. (US) 2009-06-30 US claimed