SCHEMBL4466848

SCHEMBL4466848

CCCOc1cccc(C(=O)O)c1.O=[N+]([O-])c1ccc2cccnc2c1O

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.56
MEN1 O00255 2/20 0.48
NR1H4 Q96RI1 3/20 0.47
PLA2G4B P0C869 2/20 0.45
MAPT P10636 3/20 0.43
LMNA P02545 2/20 0.43
HTT P42858 1/20 0.43
TSHR P16473 1/20 0.42
MAPK1 P28482 1/20 0.42
HSP90AA1 P07900 1/20 0.42
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
GAA P10253 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
KAT6A Q92794 1/20 0.42
PDE10A Q9Y233 1/20 0.42
TP53 P04637 1/20 0.41
POLB P06746 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4457288 0.95 PLA2G4B (0.52) KMT2AMEN1NR1H4PLA2G4BMAPT
SCHEMBL4465726 0.92 KMT2A (0.46) KMT2AMEN1NR1H4MAPTLMNA
SCHEMBL4462759 0.89 PLA2G4B (0.46) KMT2AMEN1PLA2G4BMAPTLMNA
SCHEMBL4462764 0.89 PLA2G4B (0.46) KMT2AMEN1PLA2G4BMAPTLMNA
SCHEMBL4460077 0.86 NR4A2 (0.56) NR1H4
SCHEMBL4457850 0.86 KMT2A (0.48) KMT2AMEN1MAPTLMNAHTT
M-Phenoxybenzoic Acid For Cis-Isomer SCHEMBL4460153 0.86 KDM4E (0.53) KMT2AMEN1MAPTLMNAHTT
M-Phenoxybenzoic Acid For Cis-Isomer SCHEMBL4460165 0.86 KDM4E (0.53) KMT2AMEN1MAPTLMNAHTT
SCHEMBL4461356 0.85 PLA2G4B (0.51) PLA2G4BMAPTTSHRHSP90AA1KDM4E
SCHEMBL4466851 0.83 MAPT (0.51) KMT2AMEN1MAPTLMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009140215-A2 METHOD FOR TREATING DRUG-RESISTANT BACTERIAL AND OTHER INFECTIONS WITH CLIOQUINOL, PHANQUINONE, AND RELATED COMPOUNDS GERAGHTY, ERIN (US) 2009-11-19 WO claimed
WO-2009140215-A2 METHOD FOR TREATING DRUG-RESISTANT BACTERIAL AND OTHER INFECTIONS WITH CLIOQUINOL, PHANQUINONE, AND RELATED COMPOUNDS GERAGHTY, ERIN (US) 2009-11-19 WO disclosed