SCHEMBL4457850

SCHEMBL4457850

CC(C)Oc1cccc(C(=O)O)c1.O=[N+]([O-])c1ccc2cccnc2c1O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 6/20 0.48
KDM4E B2RXH2 9/20 0.46
MAPT P10636 8/20 0.46
ALDH1A1 P00352 6/20 0.46
MEN1 O00255 4/20 0.46
GAA P10253 2/20 0.46
CTSB P07858 1/20 0.46
IDO1 P14902 1/20 0.46
TDO2 P48775 1/20 0.46
RAB9A P51151 3/20 0.44
HSP90AA1 P07900 2/20 0.44
NPC1 O15118 1/20 0.44
LMNA P02545 4/20 0.44
HTT P42858 2/20 0.44
PDE10A Q9Y233 1/20 0.43
L3MBTL1 Q9Y468 4/20 0.43
NPSR1 Q6W5P4 2/20 0.43
ADAMTS5 Q9UNA0 2/20 0.43
TDP1 Q9NUW8 1/20 0.42
HSP90AB1 P08238 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4458670 0.90 MAPT (0.51) KMT2AKDM4EMAPTALDH1A1MEN1
SCHEMBL4465726 0.88 KMT2A (0.46) KMT2AKDM4EMAPTALDH1A1MEN1
M-Phenoxybenzoic Acid For Cis-Isomer SCHEMBL4460153 0.88 KDM4E (0.53) KMT2AKDM4EMAPTALDH1A1MEN1
M-Phenoxybenzoic Acid For Cis-Isomer SCHEMBL4460165 0.88 KDM4E (0.53) KMT2AKDM4EMAPTALDH1A1MEN1
SCHEMBL4466848 0.86 KMT2A (0.56) KMT2AKDM4EMAPTALDH1A1MEN1
SCHEMBL4457288 0.85 PLA2G4B (0.52) KMT2AMAPTMEN1RAB9AHSP90AA1
SCHEMBL4460077 0.84 NR4A2 (0.56)
3,5-Dimethoxybenzoic Acid SCHEMBL4461323 0.83 EGLN1 (0.52) KMT2AKDM4EMAPTALDH1A1MEN1
3,5-Dimethoxybenzoic Acid SCHEMBL4461316 0.83 EGLN1 (0.52) KMT2AKDM4EMAPTALDH1A1MEN1
Benzoic Acid SCHEMBL4470216 0.83 ALDH1A1 (0.54) KMT2AKDM4EMAPTALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009140215-A2 METHOD FOR TREATING DRUG-RESISTANT BACTERIAL AND OTHER INFECTIONS WITH CLIOQUINOL, PHANQUINONE, AND RELATED COMPOUNDS GERAGHTY, ERIN (US) 2009-11-19 WO claimed
WO-2009140215-A2 METHOD FOR TREATING DRUG-RESISTANT BACTERIAL AND OTHER INFECTIONS WITH CLIOQUINOL, PHANQUINONE, AND RELATED COMPOUNDS GERAGHTY, ERIN (US) 2009-11-19 WO disclosed