Pamoic Acid

Pamoic Acid

SCHEMBL446833

O=C(O)c1cc2ccccc2c(Cc2c(O)c(C(=O)O)cc3ccccc23)c1O.O=C(O)c1cc2ccccc2c(Cc2c(O)c(C(=O)O)cc3ccccc23)c1O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

DRD2DRD3DRD4GNRHRHRH1HTR2AHTR2CSLC6A2SLC6A4SSTR1SSTR2SSTR3SSTR5

The experimentally established mechanism targets of Pamoic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR35 Q9HC97 2/20 1.00
POLB P06746 2/20 1.00
ME2 P23368 1/20 0.76
ME1 P48163 1/20 0.76
ME3 Q16798 1/20 0.76
MEN1 O00255 7/20 0.58
KMT2A Q03164 7/20 0.58
MAPT P10636 5/20 0.58
HPGD P15428 4/20 0.58
CYP3A4 P08684 3/20 0.58
ALOX15 P16050 3/20 0.58
MAPK1 P28482 2/20 0.58
TP53 P04637 1/20 0.58
SMN1; SMN2 Q16637 1/20 0.58
TDP1 Q9NUW8 1/20 0.58
CYP2D6 P10635 1/20 0.58
HMGB1 P09429 1/20 0.56
CXCL12 P48061 1/20 0.56
HSD17B10 Q99714 5/20 0.52
GALK1 P51570 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Pamoic Acid SCHEMBL30293211 1.00 GPR35 (1.00) GPR35POLBME2ME1ME3
Pamoic Acid SCHEMBL30293206 1.00 GPR35 (1.00) GPR35POLBME2ME1ME3
Pamoic Acid SCHEMBL5721 1.00 GPR35 (1.00) GPR35POLBME2ME1ME3
Pamoic Acid SCHEMBL29362189 1.00 GPR35 (1.00) GPR35POLBME2ME1ME3
Pamoic Acid SCHEMBL991085 0.98 GPR35 (0.97) GPR35POLBME2ME1ME3
Pamoic Acid SCHEMBL9982931 0.98 GPR35 (0.97) GPR35POLBME2ME1ME3
Pamoic Acid SCHEMBL5175194 0.98 GPR35 (0.97) GPR35POLBME2ME1ME3
Pamoic Acid SCHEMBL1055608 0.98 GPR35 (0.97) GPR35POLBME2ME1ME3
Pamoic Acid SCHEMBL5012888 0.98 GPR35 (0.97) GPR35POLBME2ME1ME3
Pamoic Acid SCHEMBL15009319 0.98 GPR35 (0.97) GPR35POLBME2ME1ME3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3347011-A1 MUSCARINIC COMBINATION AND ITS USE FOR COMBATING HYPOCHOLINERGIC DISORDERS OF THE CENTRAL NERVOUS SYSTEM Chase Pharmaceuticals Corporation (US) 2018-07-18 EP disclosed
WO-2017044693-A1 MUSCARINIC COMBINATION AND ITS USE FOR COMBATING HYPOCHOLINERGIC DISORDERS OF THE CENTRAL NERVOUS SYSTEM CHASE PHARMACEUTICALS CORPORATION (US) 2017-03-16 WO disclosed
US-20120065067-A1 PAMOIC ACID BLOCKS ETHYLENE SIGNALING THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2012-03-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120065067-A1 PAMOIC ACID BLOCKS ETHYLENE SIGNALING PAM, PRKAA1, PRKAA2 GPR35 2779/4885POLB 2224/4885ME2 395/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.