SCHEMBL4470648

SCHEMBL4470648

O=C(O)c1cccc(Br)c1.O=[N+]([O-])c1ccc2cccnc2c1O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 7/20 0.50
PDE10A Q9Y233 1/20 0.48
MAPT P10636 10/20 0.47
KDM4E B2RXH2 8/20 0.47
ALDH1A1 P00352 8/20 0.47
MEN1 O00255 5/20 0.47
IDO1 P14902 2/20 0.47
TDO2 P48775 2/20 0.47
GAA P10253 2/20 0.47
CTSB P07858 2/20 0.47
HSP90AA1 P07900 2/20 0.46
HSP90AB1 P08238 1/20 0.46
LMNA P02545 5/20 0.45
HTT P42858 3/20 0.45
L3MBTL1 Q9Y468 6/20 0.44
TDP1 Q9NUW8 4/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
PKM P14618 2/20 0.44
CASP6 P55212 2/20 0.44
POLB P06746 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4462749 0.87 RCE1 (0.55) KMT2APDE10AMAPTKDM4EALDH1A1
Benzoic Acid SCHEMBL4470216 0.87 ALDH1A1 (0.54) KMT2APDE10AMAPTKDM4EALDH1A1
Benzoic Acid SCHEMBL4470207 0.87 ALDH1A1 (0.54) KMT2APDE10AMAPTKDM4EALDH1A1
SCHEMBL4461259 0.87 ALDH1A1 (0.52) KMT2APDE10AMAPTKDM4EALDH1A1
SCHEMBL4465726 0.84 KMT2A (0.46) KMT2APDE10AMAPTKDM4EALDH1A1
M-Phenoxybenzoic Acid For Cis-Isomer SCHEMBL4460165 0.84 KDM4E (0.53) KMT2APDE10AMAPTKDM4EALDH1A1
SCHEMBL4458854 0.84 GSTP1 (0.52) KMT2APDE10AMAPTKDM4EALDH1A1
SCHEMBL4458860 0.84 GSTP1 (0.52) KMT2APDE10AMAPTKDM4EALDH1A1
M-Phenoxybenzoic Acid For Cis-Isomer SCHEMBL4460153 0.84 KDM4E (0.53) KMT2APDE10AMAPTKDM4EALDH1A1
SCHEMBL4466848 0.83 KMT2A (0.56) KMT2APDE10AMAPTKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009140215-A2 METHOD FOR TREATING DRUG-RESISTANT BACTERIAL AND OTHER INFECTIONS WITH CLIOQUINOL, PHANQUINONE, AND RELATED COMPOUNDS GERAGHTY, ERIN (US) 2009-11-19 WO claimed
WO-2009140215-A2 METHOD FOR TREATING DRUG-RESISTANT BACTERIAL AND OTHER INFECTIONS WITH CLIOQUINOL, PHANQUINONE, AND RELATED COMPOUNDS GERAGHTY, ERIN (US) 2009-11-19 WO disclosed