SCHEMBL4470693

SCHEMBL4470693

CCNC(=O)C(=O)N1CCn2cccc2C1c1ccc(C)cc1

nearest known ligand 0.58

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 7/20 0.58
MEN1 O00255 5/20 0.58
MAPT P10636 9/20 0.49
KDM4E B2RXH2 3/20 0.49
HTT P42858 3/20 0.49
ADRA2C P18825 1/20 0.48
ALDH1A1 P00352 8/20 0.48
SMN1; SMN2 Q16637 4/20 0.48
L3MBTL1 Q9Y468 2/20 0.44
GAA P10253 2/20 0.41
MAPK1 P28482 1/20 0.41
TP53 P04637 1/20 0.41
NPSR1 Q6W5P4 2/20 0.41
TDP1 Q9NUW8 1/20 0.39
RECQL P46063 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2418931 0.73 KMT2A (0.43) KMT2AMEN1MAPTKDM4EHTT
SCHEMBL1266343 0.73 ALDH1A1 (0.52) KMT2AMEN1MAPTKDM4EHTT
SCHEMBL2415540 0.72 ADRA2C (0.41) KMT2AMEN1MAPTKDM4EHTT
SCHEMBL2421577 0.72 CNR1 (0.44) KMT2AMEN1MAPTKDM4EHTT
SCHEMBL3837693 0.71 ADRA2C (0.57) KMT2AMEN1MAPTKDM4EHTT
SCHEMBL2418577 0.70 LMNA (0.50) KMT2AMEN1ALDH1A1SMN1; SMN2
SCHEMBL2419551 0.69 ALDH1A1 (0.59) KMT2AMEN1MAPTKDM4EHTT
SCHEMBL2416816 0.69 ALDH1A1 (0.55) KMT2AMEN1MAPTKDM4EHTT
SCHEMBL2418781 0.68 ALDH1A1 (0.55) KMT2AMEN1MAPTKDM4EHTT
SCHEMBL2421388 0.68 MAPT (0.41) KMT2AMEN1MAPTKDM4EHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7625900-B2 Sutstituted tetrahydropyrrolopyrazine compounds and the use thereof in the treatment and/or inhibition of pain GRUENENTHAL GMBH (DE) 2009-12-01 US claimed