SCHEMBL4472288

SCHEMBL4472288

Cc1c[c]c(N(C)CCN(C)C)cc1

nearest known ligand 0.33

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.33
CA12 O43570 1/20 0.30
CA2 P00918 1/20 0.30
CA9 Q16790 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP2D6 P10635 1/20 0.30
CYP2C19 P33261 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8660579 0.74 ALDH1A1 (0.40)
SCHEMBL28519732 0.69 ALDH1A1 (0.33)
SCHEMBL14174805 0.69 ALDH1A1 (0.50) HRH3CA12CA2CA9CYP2C19
SCHEMBL5179223 0.67 ALDH1A1 (0.34) HRH3
SCHEMBL359666 0.63 POLB (0.35)
SCHEMBL19007315 0.63 HTT (0.39) HRH3CYP1A2CYP2D6CYP2C19
SCHEMBL15872033 0.63 SMN1; SMN2 (0.46) HRH3CYP1A2CYP2D6CYP2C19
SCHEMBL27964797 0.63 ALDH1A1 (0.34) CA12CA9CYP1A2CYP2D6CYP2C19
SCHEMBL13103012 0.61 HRH3 (0.47) HRH3CYP2D6CYP2C19
SCHEMBL3707752 0.61 NOS1 (0.34) HRH3CYP2D6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7598274-B2 N-methyl-4-{4-[5-(4-chloro-3-trifluoromethylphenylcarbamoyl)-1H-pyrrol-3-yl]-phenoxy}pyridine-2-carboxamide; Raf kinases inhibitors MERCK PATENT GMBH (DE) 2009-10-06 US claimed