SCHEMBL4476392

SCHEMBL4476392

Cc1[nH]c(C)c(-c2c[nH]c(-c3ccc(C(F)(F)F)cc3C(F)(F)F)cc2=O)c(=O)c1Br

nearest known ligand 0.43

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SLC2A1 P11166 1/20 0.43
DAO P14920 1/20 0.34
MAPT P10636 1/20 0.33
TDP2 O95551 1/20 0.30
ABCC8 Q09428 1/20 0.30
KCNJ11 Q14654 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4489339 0.87 SLC2A1 (0.41) SLC2A1DAO
SCHEMBL4472791 0.87 SLC2A1 (0.46) SLC2A1DAOMAPTTDP2
SCHEMBL4493394 0.83 SLC2A1 (0.52) SLC2A1MAPT
SCHEMBL4483281 0.82 SLC2A1 (0.44) SLC2A1
SCHEMBL4491224 0.77 DAO (0.34) SLC2A1DAOMAPT
SCHEMBL4485647 0.77 HSD11B1 (0.35) SLC2A1DAOMAPT
SCHEMBL4486516 0.77 ADORA2A (0.41) SLC2A1
SCHEMBL4464654 0.76 ADORA2A (0.39) SLC2A1MAPT
SCHEMBL4476390 0.76 SLC2A1 (0.56) SLC2A1
SCHEMBL4464123 0.76 SLC2A1 (0.41) SLC2A1DAOMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7579353-B2 Pyridinone derivatives against malaria GLAXO GROUP LIMITED (GB) 2009-08-25 US claimed
US-20080287461-A1 Pyridinone Derivatives Against Malaria GLAXO GROUP LIMITED (GB) 2008-11-20 US claimed
US-7579353-B2 Pyridinone derivatives against malaria GLAXO GROUP LIMITED (GB) 2009-08-25 US disclosed
US-20080287461-A1 Pyridinone Derivatives Against Malaria GLAXO GROUP LIMITED (GB) 2008-11-20 US disclosed
EP-1858876-A2 PYRIDINONE DERIVATIVES AGAINST MALARIA GLAXO GROUP LIMITED (GB) 2007-11-28 EP disclosed
WO-2006094799-A2 PYRIDINONE DERIVATIVES AGAINST MALARIA GLAXO GROUP LIMITED (GB) 2006-09-14 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080287461-A1 Pyridinone Derivatives Against Malaria G6PD, PNPO, PLPBP SLC2A1 2278/4885DAO 2428/4885MAPT 1942/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.