SCHEMBL4476920

SCHEMBL4476920

O=S(=O)(Cl)c1c(Cl)cc(F)cc1Cl

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TRPV4 Q9HBA0 1/20 0.35
ACLY P53396 1/20 0.33
CA1 P00915 2/20 0.32
CA2 P00918 2/20 0.32
PTGS2 P35354 1/20 0.32
CA9 Q16790 1/20 0.32
PTGES2 Q9H7Z7 1/20 0.31
AKR1B1 P15121 1/20 0.31
KMT2A Q03164 1/20 0.31
CA12 O43570 1/20 0.30
CA7 P43166 1/20 0.30
CA13 Q8N1Q1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL181647 0.79 ALDH1A1 (0.43) TRPV4ACLYCA1CA2CA9
SCHEMBL20486440 0.78 CA1 (0.48) CA1CA2PTGS2CA9PTGES2
SCHEMBL1500909 0.77 CA12 (0.36) CA1CA2PTGES2CA12CA7
SCHEMBL4512524 0.75 CA1 (0.35) TRPV4CA1CA2KMT2A
SCHEMBL10958575 0.75 HSD17B10 (0.48) TRPV4CA1CA2
SCHEMBL1036314 0.75 NMT1 (0.42) TRPV4ACLYCA1CA2CA9
SCHEMBL1077563 0.75 CYP3A4 (0.48) CA1CA2CA9KMT2ACA12
SCHEMBL533215 0.75 MCL1 (0.39) KMT2A
SCHEMBL640928 0.73 PTGS1 (0.38) CA1CA2PTGS2CA9KMT2A
SCHEMBL2778353 0.73 PTGES2 (0.50) CA1CA2PTGS2CA9PTGES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023028056-A1 3-AMINO PIPERIDYL SODIUM CHANNEL INHIBITORS GENENTECH, INC. (US) 2023-03-02 WO disclosed
US-7538111-B2 Benzenesulphonamide derivatives, method for production and use thereof for treatment of pain LABORATOIRES FOURNIER S.A. (FR) 2009-05-26 US disclosed
US-20060178360-A1 Benzenesulphonamide derivatives, method for production and use thereof for treatment of pain LABORATOIRES FOURNIER S.A. (FR) 2006-08-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060178360-A1 Benzenesulphonamide derivatives, method for production and use thereof for treatment of pain LTB4R2, BDKRB2, TBXA2R TRPV4 113/4885ACLY 785/4885CA1 4375/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.