SCHEMBL4483317

SCHEMBL4483317

COc1ccc(C)cc1-c1nnc(S)n1N

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.42
CYP3A4 P08684 2/20 0.42
ACHE P22303 1/20 0.42
KDM4E B2RXH2 3/20 0.38
LMNA P02545 2/20 0.38
MDM2 Q00987 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
KMT2A Q03164 3/20 0.36
NR1I2 O75469 2/20 0.36
MAPT P10636 2/20 0.35
TSHR P16473 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2C19 P33261 1/20 0.35
BACE1 P56817 1/20 0.35
MEN1 O00255 1/20 0.34
GRM5 P41594 1/20 0.34
GAA P10253 2/20 0.34
USP2 O75604 1/20 0.34
POLB P06746 1/20 0.34
CTSA P10619 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4486268 0.88 ACHE (0.42) ALDH1A1CYP3A4ACHEKDM4ELMNA
SCHEMBL4351022 0.87 MEN1 (0.47) ALDH1A1KDM4ELMNASMN1; SMN2KMT2A
SCHEMBL4520093 0.85 ALDH1A1 (0.45) ALDH1A1KDM4ELMNASMN1; SMN2KMT2A
SCHEMBL4482344 0.85 LRRK2 (0.38) KDM4EBACE1CTSA
SCHEMBL2889816 0.81 KDM4E (0.52) ALDH1A1KDM4ELMNASMN1; SMN2KMT2A
SCHEMBL28279054 0.79 KDM4E (0.41) ALDH1A1KDM4ELMNASMN1; SMN2MAPT
SCHEMBL4346620 0.78 ALDH1A1 (0.56) ALDH1A1CYP3A4KDM4ELMNAKMT2A
SCHEMBL4341622 0.77 MAPT (0.54) ALDH1A1CYP3A4KDM4ESMN1; SMN2KMT2A
SCHEMBL4478644 0.77 KDM4E (0.39) ALDH1A1KDM4ELMNASMN1; SMN2KMT2A
SCHEMBL4342691 0.77 KDM4E (0.39) ALDH1A1KDM4EKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009094205-A2 3-ARYL-6-ARYL-7H-[1,2,4]TRIAZOLO[3,4-B][1,3,4]THIADIAZINES AND ANALOGS AS ACTIVATORS OF CASPASES AND INDUCERS OF APOPTOSIS AND THE USE THEREOF CYTOVIA, INC. (US) 2009-07-30 WO disclosed