SCHEMBL4478644

SCHEMBL4478644

COc1cc(Br)ccc1-c1nnc(S)n1N

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.39
ALDH1A1 P00352 1/20 0.39
GAA P10253 2/20 0.39
MGAM O43451 1/20 0.39
SI P14410 1/20 0.39
MGAM2 Q2M2H8 1/20 0.39
SMN1; SMN2 Q16637 4/20 0.37
LMNA P02545 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
APLNR P35414 1/20 0.37
BRD4 O60885 1/20 0.36
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
MAPK1 P28482 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
MC4R P32245 1/20 0.33
TP53 P04637 1/20 0.33
NFKB1 P19838 1/20 0.33
NFKB2 Q00653 1/20 0.33
RELA Q04206 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4486268 0.85 ACHE (0.42) KDM4EALDH1A1LMNAMEN1KMT2A
SCHEMBL4346620 0.84 ALDH1A1 (0.56) KDM4EALDH1A1GAALMNAMEN1
SCHEMBL4348022 0.83 HSP90AA1 (0.47) KDM4EALDH1A1
SCHEMBL4342691 0.83 KDM4E (0.39) KDM4EALDH1A1KMT2A
SCHEMBL4487389 0.82 MAPK14 (0.37) ALDH1A1SMN1; SMN2LMNA
SCHEMBL2889816 0.79 KDM4E (0.52) KDM4EALDH1A1SMN1; SMN2LMNAKMT2A
SCHEMBL4483317 0.77 ALDH1A1 (0.42) KDM4EALDH1A1GAASMN1; SMN2LMNA
SCHEMBL4351022 0.75 MEN1 (0.47) KDM4EALDH1A1GAASMN1; SMN2LMNA
SCHEMBL22599742 0.75 PDE2A (0.34) ALDH1A1SMN1; SMN2LMNAMEN1KMT2A
SCHEMBL25413578 0.74 ALDH1A1 (0.36) KDM4EALDH1A1GAASMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009094205-A2 3-ARYL-6-ARYL-7H-[1,2,4]TRIAZOLO[3,4-B][1,3,4]THIADIAZINES AND ANALOGS AS ACTIVATORS OF CASPASES AND INDUCERS OF APOPTOSIS AND THE USE THEREOF CYTOVIA, INC. (US) 2009-07-30 WO disclosed
WO-2009094205-A2 3-ARYL-6-ARYL-7H-[1,2,4]TRIAZOLO[3,4-B][1,3,4]THIADIAZINES AND ANALOGS AS ACTIVATORS OF CASPASES AND INDUCERS OF APOPTOSIS AND THE USE THEREOF CYTOVIA, INC. (US) 2009-07-30 WO disclosed