SCHEMBL4483879

SCHEMBL4483879

CC(=O)Nc1cccc2cc(S(=O)(=O)NCc3ccccc3)ccc12

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP6 P55212 1/20 0.64
CYP19A1 P11511 2/20 0.54
KMT2A Q03164 2/20 0.52
MEN1 O00255 1/20 0.52
PIK3CD O00329 1/20 0.52
PIK3CG P48736 1/20 0.52
POLB P06746 1/20 0.51
HDAC2 Q92769 1/20 0.49
HDAC8 Q9BY41 1/20 0.49
HDAC6 Q9UBN7 1/20 0.49
HTT P42858 1/20 0.49
SCN9A Q15858 1/20 0.48
MAPT P10636 1/20 0.48
GAA P10253 1/20 0.48
KDM4E B2RXH2 1/20 0.48
GSK3B P49841 1/20 0.48
CA12 O43570 1/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
ATM Q13315 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6906511 0.93 CASP6 (0.59) CASP6CYP19A1KMT2AMEN1PIK3CD
SCHEMBL6907200 0.91 CASP6 (0.61) CASP6CYP19A1KMT2AMEN1POLB
SCHEMBL4480386 0.88 CASP6 (0.58) CASP6CYP19A1KMT2AMEN1POLB
SCHEMBL4556308 0.86 CASP6 (0.58) CASP6CYP19A1KMT2AMEN1POLB
SCHEMBL6909638 0.86 CASP6 (0.58) CASP6CYP19A1KMT2AMEN1POLB
SCHEMBL6906323 0.85 CASP6 (0.60) CASP6CYP19A1KMT2AMEN1POLB
SCHEMBL6909319 0.84 CASP6 (0.61) CASP6CYP19A1KMT2AMEN1POLB
SCHEMBL6903974 0.84 ATM (0.64) CASP6POLBGAAATML3MBTL1
SCHEMBL4489812 0.81 LMNA (0.61) CYP19A1KMT2AMEN1PIK3CDPIK3CG
SCHEMBL4482883 0.81 CYP19A1 (0.53) CYP19A1KMT2APOLBHDAC2HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7598418-B2 Naphthalene-1-(sulfonamide or carboxamide) derivatives; e.g. N-Benzyl-5-{[(4-methylphenyl)sulfonyl]oxy}naphthalene-1-sulfonamide; protein kinase inhibitors sensitize cancer cells to radiotherapy or anticancer agents; side effect reduction INSTITUTE OF MEDICINAL MOLECULAR DESIGN, INC. (JP) 2009-10-06 US claimed
US-20050215645-A1 Amide derivatives INSTITUTE OF MEDICINAL MOLECULAR DESIGN. INC. (JP) 2005-09-29 US claimed
US-7598418-B2 Naphthalene-1-(sulfonamide or carboxamide) derivatives; e.g. N-Benzyl-5-{[(4-methylphenyl)sulfonyl]oxy}naphthalene-1-sulfonamide; protein kinase inhibitors sensitize cancer cells to radiotherapy or anticancer agents; side effect reduction INSTITUTE OF MEDICINAL MOLECULAR DESIGN, INC. (JP) 2009-10-06 US disclosed
US-20050215645-A1 Amide derivatives INSTITUTE OF MEDICINAL MOLECULAR DESIGN. INC. (JP) 2005-09-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050215645-A1 Amide derivatives OGG1, HDAC1, BCL2A1 CASP6 381/4885CYP19A1 552/4885KMT2A 1012/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.