SCHEMBL4486435

SCHEMBL4486435

CCC(=O)Nc1n[nH]c2cc(-c3ccsc3)ccc12

nearest known ligand 0.85

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 19/20 0.85
CYP1A2 P05177 3/20 0.85
CDK2 P24941 1/20 0.72
GSK3A P49840 1/20 0.72
HDAC1 Q13547 1/20 0.72
HDAC2 Q92769 1/20 0.72
HDAC8 Q9BY41 1/20 0.72

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1462380 0.92 GSK3B (1.00) GSK3BCYP1A2CDK2GSK3AHDAC1
SCHEMBL4487631 0.87 GSK3B (0.75) GSK3BCYP1A2CDK2GSK3AHDAC1
SCHEMBL4486330 0.84 GSK3B (0.75) GSK3BCYP1A2CDK2GSK3AHDAC1
SCHEMBL4497828 0.84 GSK3B (1.00) GSK3BCYP1A2CDK2GSK3AHDAC1
SCHEMBL4493554 0.84 GSK3B (0.71) GSK3BCYP1A2CDK2GSK3AHDAC1
SCHEMBL4489321 0.83 GSK3B (0.76) GSK3BCYP1A2
SCHEMBL4487680 0.83 GSK3B (0.84) GSK3BCYP1A2GSK3AHDAC1HDAC2
SCHEMBL4492445 0.83 GSK3B (0.70) GSK3BCYP1A2CDK2GSK3AHDAC1
SCHEMBL4483246 0.82 GSK3B (0.69) GSK3BCYP1A2CDK2GSK3AHDAC1
SCHEMBL4483590 0.82 GSK3B (0.84) GSK3BCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7632854-B2 Aminoindazole derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions comprising them PFIZER ITALIA S.R.L. (IT) 2009-12-15 US claimed