SCHEMBL4493399

SCHEMBL4493399

CC[C@@H](C(N)=O)N1C[C@@H](CO)CCC1=O

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.55
CA12 O43570 1/20 0.55
CA1 P00915 1/20 0.55
CA2 P00918 1/20 0.55
CA3 P07451 1/20 0.55
CA4 P22748 1/20 0.55
CA6 P23280 1/20 0.55
CA5A P35218 1/20 0.55
CA7 P43166 1/20 0.55
CA9 Q16790 1/20 0.55
CA13 Q8N1Q1 1/20 0.55
CA14 Q9ULX7 1/20 0.55
CA5B Q9Y2D0 1/20 0.55
BRD4 O60885 1/20 0.36
LIPE Q05469 1/20 0.30
P2RX7 Q99572 1/20 0.30
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL661204 1.00 LMNA (0.55) LMNACA12CA1CA2CA3
SCHEMBL4507352 1.00 LMNA (0.55) LMNACA12CA1CA2CA3
SCHEMBL4500199 1.00 LMNA (0.55) LMNACA12CA1CA2CA3
SCHEMBL660725 0.92 LMNA (0.60) LMNACA12CA1CA2CA3
SCHEMBL661497 0.90 LMNA (0.61) LMNACA12CA1CA2CA3
SCHEMBL663106 0.87 LMNA (0.54) LMNACA12CA1CA2CA3
SCHEMBL661034 0.87 LMNA (0.54) LMNACA12CA1CA2CA3
SCHEMBL661877 0.87 LMNA (0.54) LMNACA12CA1CA2CA3
SCHEMBL660117 0.87 LMNA (0.54) LMNACA12CA1CA2CA3
SCHEMBL28176514 0.86 LMNA (0.52) LMNACA12CA1CA2CA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20060258704-A1 2-Oxo-piperidinyl- and 2-oxo-azepanyl alkanoic acid derivatives for the treatment of epilepsy and other neurological disorders MICHEL PHILIPPE 2006-11-16 US claimed
US-20040132717-A1 2-Oxo-piperidinyl-and 2-oxo-azepanyl alkanoic acid derivatives for the treatment of epilepsy and other neurological disorders UCB, S.A. (BE) 2004-07-08 US claimed
EP-1395560-A1 2-OXO-PIPERIDINYL- AND 2-OXO-AZEPANYL ALKANOIC ACID DERIVATIV ES FOR THE TREATMENT OF EPILEPSY AND OTHER NEUROLOGICAL DISORDERS UCB, S.A. (BE) 2004-03-10 EP claimed
WO-2002094787-A1 2-OXO-PIPERIDINYL- AND 2-OXO-AZEPANYL ALKANOIC ACID DERIVATIV ES FOR THE TREATMENT OF EPILEPSY AND OTHER NEUROLOGICAL DISORDERS UCB, S.A. (BE) 2002-11-28 WO claimed
US-7473697-B2 2-Oxo-piperidinyl- and 2-oxo-azepanyl alkanoic acid derivatives for the treatment of epilepsy and other neurological disorders UCB S.A. (BE) 2009-01-06 US disclosed
US-20060258704-A1 2-Oxo-piperidinyl- and 2-oxo-azepanyl alkanoic acid derivatives for the treatment of epilepsy and other neurological disorders MICHEL PHILIPPE 2006-11-16 US disclosed
US-7087596-B2 2-oxo-piperidinyl- and 2-oxo-azepanyl alkanoic acid derivatives for the treatment of epilepsy and other neurological disorders UCB, S.A. (BE) 2006-08-08 US disclosed
US-20040132717-A1 2-Oxo-piperidinyl-and 2-oxo-azepanyl alkanoic acid derivatives for the treatment of epilepsy and other neurological disorders UCB, S.A. (BE) 2004-07-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040132717-A1 2-Oxo-piperidinyl-and 2-oxo-azepanyl alkanoic acid derivatives for the treatment of epilepsy and other neurological disorders GABRA6, GABRA2, HCAR2 LMNA 2596/4885CA12 2989/4885CA1 723/4885
US-20060258704-A1 2-Oxo-piperidinyl- and 2-oxo-azepanyl alkanoic acid derivatives for the treatment of epilepsy and other neurological disorders GABRA6, HCAR2, GABRA2 LMNA 2587/4885CA12 2982/4885CA1 764/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.