SCHEMBL45056

SCHEMBL45056

CCCCCOCC(O)COP(=O)(O)O

nearest known ligand 0.97

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
LPAR5 Q9H1C0 6/20 0.97
LPAR1 Q92633 13/20 0.67
LPAR3 Q9UBY5 10/20 0.67
LPAR2 Q9HBW0 7/20 0.59
LPAR4 Q99677 5/20 0.59
LPAR6 P43657 4/20 0.59
ENPP2 Q13822 3/20 0.59
USP2 O75604 1/20 0.56
HTT P42858 1/20 0.54
P2RY10 O00398 1/20 0.54
CES2 O00748 1/20 0.51
TRPV1 Q8NER1 1/20 0.51
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2C19 P33261 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL250888 1.00 LPAR5 (0.97) LPAR5LPAR1LPAR3LPAR2LPAR4
SCHEMBL258161 0.98 LPAR5 (1.00) LPAR5LPAR1LPAR3LPAR2LPAR4
SCHEMBL7820593 0.98 LPAR5 (1.00) LPAR5LPAR1LPAR3LPAR2LPAR4
SCHEMBL258032 0.98 LPAR5 (1.00) LPAR5LPAR1LPAR3LPAR2LPAR4
SCHEMBL258118 0.98 LPAR5 (1.00) LPAR5LPAR1LPAR3LPAR2LPAR4
SCHEMBL7829804 0.98 LPAR5 (1.00) LPAR5LPAR1LPAR3LPAR2LPAR4
SCHEMBL12621099 0.98 LPAR5 (1.00) LPAR5LPAR1LPAR3LPAR2LPAR4
SCHEMBL258094 0.98 LPAR5 (1.00) LPAR5LPAR1LPAR3LPAR2LPAR4
SCHEMBL28064781 0.98 LPAR5 (1.00) LPAR5LPAR1LPAR3LPAR2LPAR4
SCHEMBL26603866 0.98 LPAR5 (1.00) LPAR5LPAR1LPAR3LPAR2LPAR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 56 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111154724-A Extracted plant lipids comprising docosahexaenoic acid 联邦科学技术研究组织 2020-05-15 CN claimed
US-20120270250-A1 TEST SYSTEM FOR MEASURING MEST ACTIVITY AS WELL AS METHODS AND USES INVOLVING THE SAME SANOFI (FR) 2012-10-25 US claimed
EP-2446050-A1 TEST SYSTEM FOR MEASURING MEST ACTIVITY AS WELL AS METHODS AND USES INVOLVING THE SAME SANOFI (FR) 2012-05-02 EP claimed
EP-2283137-A1 RECOMBINANT CELLS AND METHODS FOR HYDROXYLATING FATTY ACIDS Commonwealth Scientific and Industrial Research Organisation (AU) 2011-02-16 EP claimed
WO-2010149780-A1 TEST SYSTEM FOR MEASURING MEST ACTIVITY AS WELL AS METHODS AND USES INVOLVING THE SAME SANOFI-AVENTIS (FR) 2010-12-29 WO claimed
EP-2267152-A1 Test system for measuring MEST activity as well as methods and uses involving the same Sanofi-Aventis (FR) 2010-12-29 EP claimed
WO-2009129582-A1 POLYPEPTIDES AND METHODS FOR PRODUCING TRIACYLGLYCEROLS COMPRISING MODIFIED FATTY ACIDS COMMONWEALTH SCIENTIFIC INDUSTRIAL RESEARCH ORGANISATION (AU) 2009-10-29 WO claimed
WO-2009129583-A1 RECOMBINANT CELLS AND METHODS FOR HYDROXYLATING FATTY ACIDS COMMONWEALTH SCIENTIFIC INDUSTRIAL RESEARCH ORGANISATION (AU) 2009-10-29 WO claimed
EP-1615937-A2 ANALOGS OF LYSOPHOSPHATIDIC ACID AND METHODS OF MAKING AND USING THEREOF University of Utah Research Foundation (US) 2006-01-18 EP claimed
WO-2004092188-A2 ANALOGS OF LYSOPHOSPHATIDIC ACID AND METHODS OF MAKING AND USING THEREOF UNIVERSITY OF UTAH RESEARCH FOUNDATION (US) 2004-10-28 WO claimed
US-5827831-A Lipid nucleotide analog prodrugs for oral administration NEXSTAR PHARMACEUTICALS, INC. (US) 1998-10-27 US claimed
WO-2023141470-A2 IMMUNOMODULATORY LIPIDS AND USES THEREOF PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2023-07-27 WO disclosed
WO-2023102425-A1 METHODS FOR DETERMINING OPIOID RESPONSIVENESS IN THE TREATMENT OF PAIN EAST CAROLINA UNIVERSITY (US) 2023-06-08 WO disclosed
US-20170211013-A1 LIPID COMPRISING LONG CHAIN POLYUNSATURATED FATTY ACIDS COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2017-07-27 US disclosed
US-20170088842-A1 GENETICALLY MODIFIED FUNGI AND THEIR USE IN LIPID PRODUCTION TEKNOLOGIAN TUTKIMUSKESKUS VTT (FI) 2017-03-30 US disclosed
EP-1278858-A2 46743 AND 27417, NOVEL HUMAN ACYLTRANSFERASE FAMILY MEMBERS AND USES THEREFOR Millennium Pharmaceuticals, Inc. (US) 2003-01-29 EP disclosed
US-20020016449-A1 46743 and 27417, novel human acyltransferase family members and uses therefor MILLENNIUM PHARMACEUTICALS, INC. 2002-02-07 US disclosed
US-20020007499-A1 DNA SEQUENCE ENCODING PLANT 2-ACYLTRANSFERASE GENE SHEARS PTY. LIMITED (AU) 2002-01-17 US disclosed
WO-2001073051-A2 46743 AND 27417, NOVEL HUMAN ACYLTRANSFERASE FAMILY MEMBERS AND USES THEREFOR MILLENNIUM PHARMACEUTICALS, INC. (US) 2001-10-04 WO disclosed
US-6210967-B1 NUCLEOTIDE SEQUENCES CODING HUMAN PHOSPHATIDIC ACID BINDING PROTEIN; FOR TREATMENT AND PREVENTION OF CANCER, PLATELET AGGREGATION, VASCULAR RESTENOSIS, ARTHRITIS, WOUND HEALING, TISSUE REGENERATION, COAGULATION, OSTEOPOROSIS AND SCARING SYNAPTIC PHARMACEUTICAL CORPORATION 2001-04-03 US disclosed