SCHEMBL4507481

SCHEMBL4507481

CSc1ccccc1Cn1c(C)cc(OCc2ccccc2CNC(N)=O)c(Cl)c1=O

nearest known ligand 0.46

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 14/20 0.46
LMNA P02545 2/20 0.35
MAPT P10636 2/20 0.34
L3MBTL1 Q9Y468 2/20 0.34
ALDH1A1 P00352 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4521648 0.91 MAPK14 (0.43) MAPK14LMNAMAPTL3MBTL1ALDH1A1
SCHEMBL4504769 0.87 MAPK14 (0.49) MAPK14MAPTALDH1A1MEN1KMT2A
SCHEMBL4517123 0.86 MAPK14 (0.51) MAPK14LMNAMAPTALDH1A1KMT2A
SCHEMBL4512169 0.84 MAPK14 (0.52) MAPK14MAPT
SCHEMBL4504766 0.82 MAPK14 (0.40) MAPK14LMNAMAPTALDH1A1MEN1
SCHEMBL4508090 0.81 MAPK14 (0.50) MAPK14MAPTKMT2A
SCHEMBL4515517 0.81 MAPK14 (0.48) MAPK14MAPTALDH1A1
SCHEMBL4513949 0.81 MAPK14 (0.50) MAPK14MAPTKMT2A
SCHEMBL14435153 0.81 MAPK14 (0.40) MAPK14LMNAMAPTALDH1A1KMT2A
SCHEMBL4511761 0.78 MAPK14 (0.52) MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090270350-A1 Pyridinone Pyrazole Urea and Pyrimidinone Pyrazole Urea Derivatives PFIZER INC. 2009-10-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090270350-A1 Pyridinone Pyrazole Urea and Pyrimidinone Pyrazole Urea Derivatives PDXK, UMPS, CDK2 MAPK14 117/4885LMNA 2954/4885MAPT 2264/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.