SCHEMBL4508734

SCHEMBL4508734

O=C(C(=CCl)c1ccccc1)N1CCC(c2ccccc2)CC1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.52
HPGD P15428 5/20 0.51
MEN1 O00255 2/20 0.51
KMT2A Q03164 2/20 0.51
ALDH1A1 P00352 1/20 0.51
LMNA P02545 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51
SLC18A3 Q16572 1/20 0.48
BACE1 P56817 1/20 0.48
SIGMAR1 Q99720 1/20 0.48
CA12 O43570 1/20 0.47
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
CA7 P43166 1/20 0.47
CA9 Q16790 1/20 0.47
CA14 Q9ULX7 1/20 0.47
HSD11B1 P28845 1/20 0.47
KCNH2 Q12809 1/20 0.47
HRH3 Q9Y5N1 1/20 0.47
NPC1 O15118 3/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2903223 0.81 SIGMAR1 (0.47) IDO1HPGDKMT2AALDH1A1LMNA
SCHEMBL4206605 0.77 CA12 (0.71) HPGDMEN1KMT2AALDH1A1SLC18A3
SCHEMBL13589641 0.75 HRH3 (0.57) IDO1ALDH1A1SLC18A3BACE1CA12
SCHEMBL1193744 0.75 KCNH2 (0.56) IDO1HPGDALDH1A1LMNASLC18A3
SCHEMBL27888979 0.74 KCNH2 (0.73) IDO1HPGDALDH1A1SLC18A3BACE1
SCHEMBL1531725 0.74 KCNH2 (0.59) IDO1HPGDALDH1A1SLC18A3BACE1
SCHEMBL19988362 0.73 HTR2B (0.64) IDO1ALDH1A1BACE1CA12CA1
SCHEMBL10720211 0.73 CA12 (0.76) MEN1KMT2AALDH1A1SLC18A3CA12
Hydrogen Sulfide SCHEMBL27863722 0.73 KCNH2 (0.58) IDO1HPGDALDH1A1SLC18A3BACE1
SCHEMBL10720101 0.73 PARP14 (0.65) ALDH1A1LMNASLC18A3CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7632829-B2 Diazepan derivatives HOFFMANN-LA ROCHE INC. (US) 2009-12-15 US disclosed
US-20070249589-A1 Novel diazepan derivatives F. HOFFMANN-LA ROCHE AG, A SWISS COMPANY (CH) 2007-10-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070249589-A1 Novel diazepan derivatives CCR3, CCR1, CCR10 IDO1 988/4885HPGD 2904/4885MEN1 2072/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.