SCHEMBL2903223

SCHEMBL2903223

O=C1CCN(C(=O)C(=CCl)c2ccccc2)CCN1CCN1CCC(c2ccccc2)CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.47
SLC18A3 Q16572 2/20 0.42
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41
GAA P10253 1/20 0.41
KMT2A Q03164 1/20 0.41
HTR1A P08908 1/20 0.41
ADRA1B P35368 1/20 0.41
DRD2 P14416 3/20 0.40
CARM1 Q86X55 1/20 0.40
PRMT6 Q96LA8 1/20 0.40
MCHR1 Q99705 1/20 0.40
CHRM2 P08172 2/20 0.39
CHRM4 P08173 2/20 0.39
CHRM5 P08912 2/20 0.39
CHRM1 P11229 2/20 0.39
CHRM3 P20309 2/20 0.39
DRD4 P21917 1/20 0.39
DRD3 P35462 1/20 0.39
CCR5 P51681 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4508734 0.81 IDO1 (0.52) SIGMAR1SLC18A3ALDH1A1LMNAKMT2A
SCHEMBL2903219 0.76 MAPT (0.51) SIGMAR1SLC18A3ALDH1A1LMNAKMT2A
SCHEMBL2903225 0.75 ALDH1A1 (0.54) ALDH1A1LMNAKMT2ADRD2DRD3
SCHEMBL2903456 0.70 CCR2 (0.51) ALDH1A1LMNAKMT2ADRD2DRD3
SCHEMBL2903457 0.70 CCR2 (0.51) ALDH1A1LMNAKMT2ADRD2DRD3
SCHEMBL4509129 0.69 DRD2 (0.50) SIGMAR1SLC18A3KMT2AHTR1AADRA1B
SCHEMBL2903643 0.69 CCR2 (0.61)
SCHEMBL2903645 0.69 CCR2 (0.61)
SCHEMBL14587419 0.66 SIGMAR1 (1.00) SIGMAR1SLC18A3ALDH1A1LMNAGAA
SCHEMBL2904849 0.64 MEN1 (0.58) ALDH1A1LMNAGAAKMT2AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010506-B1 DIAZEPAN DERIVATIVES MODULATORS OF CHEMOKINE RECEPTORS HOFFMANN LA ROCHE (CH) 2010-08-04 EP disclosed