SCHEMBL4511967

SCHEMBL4511967

O=C1CCN(CC2CO2)CCN1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.42
HBB P68871 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
LTA4H P09960 2/20 0.42
LMNA P02545 1/20 0.39
PKM P14618 1/20 0.39
CRBN Q96SW2 2/20 0.33
OR51E2 Q9H255 1/20 0.33
MAPT P10636 1/20 0.33
POLB P06746 3/20 0.33
DHFR P00374 1/20 0.33
FKBP5 Q13451 1/20 0.32
GLA P06280 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
KDM4E B2RXH2 4/20 0.31
GAA P10253 1/20 0.31
ALDH1A1 P00352 1/20 0.31
CDA P32320 1/20 0.31
TOP2A P11388 1/20 0.30
TOP2B Q02880 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7568260 0.73 SMN1; SMN2 (0.39) TP53HBBSMN1; SMN2LMNAPOLB
SCHEMBL774001 0.72 CRBN (0.40) SMN1; SMN2LTA4HLMNAPKMCRBN
SCHEMBL14107874 0.72 CRBN (0.40) LTA4HLMNAPKMCRBNOR51E2
SCHEMBL17599183 0.71 SMN1; SMN2 (0.48) TP53HBBSMN1; SMN2MAPTPOLB
SCHEMBL4498693 0.71 OR51E2 (0.43) LTA4HLMNAPKMCRBNOR51E2
SCHEMBL3211746 0.70
SCHEMBL354055 0.70 TP53 (0.48) TP53HBBSMN1; SMN2MAPTDHFR
SCHEMBL14941658 0.69 LMNA (0.38) SMN1; SMN2LTA4HLMNAPKMCRBN
SCHEMBL15333289 0.69 LMNA (0.38) SMN1; SMN2LTA4HLMNAPKMCRBN
SCHEMBL24405214 0.68 ADRA2A (0.35) LTA4HDHFRGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7632829-B2 Diazepan derivatives HOFFMANN-LA ROCHE INC. (US) 2009-12-15 US disclosed
US-20070249589-A1 Novel diazepan derivatives F. HOFFMANN-LA ROCHE AG, A SWISS COMPANY (CH) 2007-10-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070249589-A1 Novel diazepan derivatives CCR3, CCR1, CCR10 TP53 4853/4885HBB 4305/4885SMN1; SMN2 2573/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.