Pumaprazole

Pumaprazole

SCHEMBL451376

COC(=O)Nc1cccc(C)c1CNc1cccn2c(C)c(C)nc12

nearest known ligand 0.69

Full drug profile on Sugi Atlas →

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 19/20 0.69
CYP2C9 P11712 19/20 0.69
CYP2D6 P10635 11/20 0.69
CYP2C19 P33261 9/20 0.69
CYP1A2 P05177 8/20 0.69

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Pumaprazole SCHEMBL29493303 1.00 CYP3A4 (0.69) CYP3A4CYP2C9CYP2D6CYP2C19CYP1A2
SCHEMBL1812546 0.93 CYP3A4 (0.68) CYP3A4CYP2C9CYP2D6CYP2C19CYP1A2
SCHEMBL1812877 0.91 CYP3A4 (0.60) CYP3A4CYP2C9CYP2D6CYP2C19CYP1A2
SCHEMBL1817519 0.91 CYP3A4 (0.62) CYP3A4CYP2C9CYP2D6CYP2C19CYP1A2
SCHEMBL1812857 0.91 CYP3A4 (0.62) CYP3A4CYP2C9CYP2D6CYP2C19CYP1A2
SCHEMBL9099268 0.90 CYP3A4 (0.55) CYP3A4CYP2C9CYP2D6CYP2C19CYP1A2
SCHEMBL9097344 0.89 CYP3A4 (0.54) CYP3A4CYP2C9CYP2D6CYP2C19CYP1A2
SCHEMBL1816283 0.89 CYP3A4 (0.54) CYP3A4CYP2C9CYP2D6CYP2C19CYP1A2
SCHEMBL7503350 0.89 CYP3A4 (0.60) CYP3A4CYP2C9CYP2D6CYP2C19CYP1A2
Hydrochloric Acid SCHEMBL6381033 0.89 CYP3A4 (0.60) CYP3A4CYP2C9CYP2D6CYP2C19CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 533 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111249250-A Oral capsule for treating helicobacter pylori infection 上海理工大学 2020-06-09 CN claimed
US-10130618-B2 Pharmaceutical combinations of dabigatran and proton pump inhibitors SANOVEL ILAC SANAYI VE TICARET ANONIM SIRKETI (TR) 2018-11-20 US claimed
US-20170035745-A1 PHARMACEUTICAL COMBINATIONS OF DABIGATRAN AND PROTON PUMP INHIBITORS SANOVEL ILAC SANAYI VE TICARET ANONIM SIRKETI (TR) 2017-02-09 US claimed
EP-2933002-A1 PHARMACEUTICAL COMBINATIONS OF DABIGATRAN AND PROTON PUMP INHIBITORS Sanovel Ilac Sanayi ve Ticaret A.S. (TR) 2015-10-21 EP claimed
WO-2015155281-A1 PHARMACEUTICAL COMBINATIONS OF DABIGATRAN AND PROTON PUMP INHIBITORS SANOVEL ILAC SANAYI VE TICARET A.S. (TR) 2015-10-15 WO claimed
WO-2015155307-A1 PHARMACEUTICAL COMBINATIONS OF RIVAROXABAN AND PROTON PUMP INHIBITORS SANOVEL ILAC SANAYI VE TICARET A.S. (TR) 2015-10-15 WO claimed
EP-2929885-A1 PHARMACEUTICAL COMBINATIONS OF RIVAROXABAN AND PROTON PUMP INHIBITORS Sanovel Ilac Sanayi ve Ticaret A.S. (TR) 2015-10-14 EP claimed
US-9016221-B2 Surface topographies for non-toxic bioadhesion control UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2015-04-28 US claimed
US-20150086497-A1 Skin Lightening Compositions ELC MAN LLC (US) 2015-03-26 US claimed
US-20130078305-A1 Pharmaceutical Compositions For The Coordinated Delivery Of NSAIDs POZEN, INC. (US) 2013-03-28 US claimed
CN-1147292-C Double capsule for the administration of active principles in multiple therepies ������ҩ�����޹�˾ 2004-04-28 CN claimed
EP-1336602-A1 Nitrate prodrugs able to release nitric oxide in a controlled and selective way and their use for prevention and treatment of inflammatory, ischemic and proliferative diseases Scaramuzzino, Giovanni (IT) 2003-08-20 EP claimed
EP-0841904-B1 ORAL PHARMACEUTICAL COMPOSITIONS WITH DELAYED RELEASE OF REVERSIBLE PROTON PUMP INHIBITORS ALTANA PHARMA AG (DE) 2003-02-05 EP claimed
US-6132768-A FOR TREATING DISORDERS CAUSED BY HELICOBACTER BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 2000-10-17 US claimed
EP-0683780-B1 IMIDAZOPYRIDINES AND THEIR USE IN TREATING GASTROINTESTINAL DISEASES BYK GULDEN LOMBERG CHEM FAB (DE) 2000-04-26 EP claimed
EP-0841904-A1 ORAL PHARMACEUTICAL COMPOSITIONS WITH DELAYED RELEASE OF REVERSIBLE PROTON PUMP INHIBITORS Byk Gulden Lomberg Chemische Fabrik GmbH (DE) 1998-05-20 EP claimed
US-5665730-A GASTROINTESTINAL DISORDERS BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1997-09-09 US claimed
WO-1997002021-A1 ORAL PHARMACEUTICAL COMPOSITIONS WITH DELAYED RELEASE OF REVERSIBLE PROTON PUMP INHIBITORS BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1997-01-23 WO claimed
EP-0683780-A1 IMIDAZOPYRIDINES AND THEIR USE IN TREATING GASTROINTESTINAL DISEASES Byk Gulden Lomberg Chemische Fabrik GmbH (DE) 1995-11-29 EP claimed
WO-1994018199-A1 IMIDAZOPYRIDINES AND THEIR USE IN TREATING GASTROINTESTINAL DISEASES BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1994-08-18 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170035745-A1 PHARMACEUTICAL COMBINATIONS OF DABIGATRAN AND PROTON PUMP INHIBITORS ABCB11, SLC9A5, SLC9A3 CYP3A4 70/4885CYP2C9 20/4885CYP2D6 18/4885
US-10130618-B2 Pharmaceutical combinations of dabigatran and proton pump inhibitors ABCB11, SLC9A5, SLC9A3 CYP3A4 70/4885CYP2C9 20/4885CYP2D6 18/4885
US-20150086497-A1 Skin Lightening Compositions CUTA, TYR, DSG1 CYP3A4 2827/4885CYP2C9 2552/4885CYP2D6 2870/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.