SCHEMBL4518803

SCHEMBL4518803

Cc1cccnc1CN(Cc1ncccc1C)C1CCN(C(=O)ON)CC1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 1/20 0.41
GRIN2B Q13224 4/20 0.40
CCR5 P51681 2/20 0.39
CXCR4 P61073 1/20 0.39
TDP1 Q9NUW8 1/20 0.38
KMT2A Q03164 2/20 0.38
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
KCNH2 Q12809 1/20 0.37
CHRM4 P08173 1/20 0.37
FAAH O00519 1/20 0.36
MGLL Q99685 1/20 0.36
SSTR4 P31391 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12935360 0.87 CCR5 (0.41) CCR5CXCR4TDP1KMT2AMEN1
SCHEMBL2084788 0.87 NOS2 (0.43) NOS2GRIN2BCCR5CXCR4KMT2A
SCHEMBL2082179 0.87 GPR119 (0.51) KMT2AMEN1
SCHEMBL2084919 0.86 TDP1 (0.42) NOS2GRIN2BCCR5CXCR4TDP1
Hydroxyamine SCHEMBL4518793 0.86 CCR5 (0.43) GRIN2BCCR5CXCR4TDP1KMT2A
SCHEMBL4535370 0.86 CCR5 (0.44) NOS2CCR5CXCR4TDP1KMT2A
SCHEMBL2081000 0.86 TDP1 (0.47) CCR5CXCR4TDP1KCNH2
SCHEMBL2082352 0.85 SMO (0.43) GRIN2BCCR5CXCR4TDP1KMT2A
SCHEMBL2086100 0.84 TRPV1 (0.42) NOS2GRIN2BCCR5CXCR4TDP1
SCHEMBL2083744 0.84 BTK (0.43) CCR5CXCR4TDP1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1613613-A4 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2009-03-25 EP disclosed
US-7291631-B2 CXCR4 chemokine receptor binding compounds GENZYME CORPORATION (US) 2007-11-06 US disclosed
EP-1613613-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-01-11 EP disclosed
WO-2004091518-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2004-10-28 WO disclosed