SCHEMBL4523110

SCHEMBL4523110

CC1[C@H](N)C(=O)N1S(=O)(=O)O

nearest known ligand 0.36

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
FAP Q12884 1/20 0.30
USP2 O75604 1/20 0.30
ESR1 P03372 1/20 0.30
AADAT Q8N5Z0 1/20 0.30
KDM4E B2RXH2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7811435 1.00 FAP (0.30) FAPUSP2ESR1AADATKDM4E
SCHEMBL8311603 1.00 FAP (0.30) FAPUSP2ESR1AADATKDM4E
SCHEMBL9486743 1.00 FAP (0.30) FAPUSP2ESR1AADATKDM4E
SCHEMBL8311599 1.00 FAP (0.30) FAPUSP2ESR1AADATKDM4E
SCHEMBL7811433 1.00 FAP (0.30) FAPUSP2ESR1AADATKDM4E
SCHEMBL1686983 1.00 FAP (0.30) FAPUSP2ESR1AADATKDM4E
SCHEMBL22582139 0.96 USP2 (0.31) USP2ESR1KDM4E
SCHEMBL16673765 0.77
SCHEMBL19486294 0.74
SCHEMBL9470709 0.74 USP2 (0.37) USP2ESR1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 40 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110372248-B Preparation method of anti-mud agent suitable for high-mud-content concrete 北京工业大学 2021-08-13 CN claimed
CN-109761871-B Synthetic method of aztreonam monocyclic parent nucleus 山东昌邑四方医药化工有限公司 2020-11-24 CN claimed
US-7601832-B2 combining [3S]3-amino-4-methyl-2-oxo-1-azetidinesulfonic acid with TAEM to obtain [3S-[3 alpha (Z),4 beta ]]-3-[[(2-amino-4-thiazolyl)[(1-carboxy-1-methylethoxy)imino]acetyl]amino]-4-methyl-2-oxo-1-azetidinesulfonic acid; one pot processs; antibiotic SICOR, INC. (US) 2009-10-13 US claimed
CN-110372248-B Preparation method of anti-mud agent suitable for high-mud-content concrete 北京工业大学 2021-08-13 CN disclosed
CN-110372248-B Preparation method of anti-mud agent suitable for high-mud-content concrete 北京工业大学 2021-08-13 CN disclosed
CN-109761871-B Synthetic method of aztreonam monocyclic parent nucleus 山东昌邑四方医药化工有限公司 2020-11-24 CN disclosed
CN-100586930-C Preparation method of aztreonam intermediate (3S-trans)-3-amido-4-methyl-2-oxo-1-sulfoazetidine CHONGQING LUMMY PHARMACEUTICAL 2010-02-03 CN disclosed
US-7601832-B2 combining [3S]3-amino-4-methyl-2-oxo-1-azetidinesulfonic acid with TAEM to obtain [3S-[3 alpha (Z),4 beta ]]-3-[[(2-amino-4-thiazolyl)[(1-carboxy-1-methylethoxy)imino]acetyl]amino]-4-methyl-2-oxo-1-azetidinesulfonic acid; one pot processs; antibiotic SICOR, INC. (US) 2009-10-13 US disclosed
US-7601832-B2 combining [3S]3-amino-4-methyl-2-oxo-1-azetidinesulfonic acid with TAEM to obtain [3S-[3 alpha (Z),4 beta ]]-3-[[(2-amino-4-thiazolyl)[(1-carboxy-1-methylethoxy)imino]acetyl]amino]-4-methyl-2-oxo-1-azetidinesulfonic acid; one pot processs; antibiotic SICOR, INC. (US) 2009-10-13 US disclosed
CN-101362713-A Preparation method of (3S-trans)-3-amido-4-methyl-2-oxo-1-sulfoazetidine CHONGQING LUMMY PHARMACEUTICAL (CN) 2009-02-11 CN disclosed
US-6916803-B2 3-(Heteroaryl acetamido)-2-oxo-azetidine-1-sulfonic acids derivatives as antibacterial agents PANTHERIX, LTD. (GB) 2005-07-12 US disclosed
US-4596777-A Process for preparing (3S)-3-[[[2-(protected or unprotected amino)-4-thiazolyl]acetyl]amino]-2-oxo-1-azetidinesulfonic acid and 4-substituted derivatives thereof E. R. SQUIBB & SONS, INC. (US) 1986-06-24 US disclosed
EP-0086556-B1 PROCESS FOR PREPARING (3S)-3-(((2-AMINO-4-THIAZOLYL)((1-CARBOXY-1-METHYLETHOXY)IMINO)-ACETYL)AMINO)-2-OXO-1-AZETIDINESULFONIC ACID AND 4-SUBSTITUTED DERIVATIVES E.R. Squibb & Sons, Inc. (US) 1986-05-07 EP disclosed
US-4529698-A Culturing Chromobacterium E. R. SQUIBB & SONS, INC. (US) 1985-07-16 US disclosed
US-4483797-A (S)-3-Isocyanato-2-oxo-1-azetidinesulfonic acids E. R. SQUIBB & SONS, INC. (US) 1984-11-20 US disclosed
US-4443374-A Process for preparing (3S)-3-[[(2-amino-4-thiazolyl)[(1-carboxy-1-methylethoxy)imino]-acetyl]amino]-2-oxo-1-azetidinesulfonic acid, and 4-substituted derivatives E. R. SQUIBB & SONS, INC. (US) 1984-04-17 US disclosed
EP-0097352-A2 Process for the preparation of azetidine sulfonic acids E.R. Squibb & Sons, Inc. (US) 1984-01-04 EP disclosed
EP-0086556-A1 Process for preparing (3S)-3-(((2-amino-4-thiazolyl)((1-carboxy-1-methylethoxy)imino)-acetyl)amino)-2-oxo-1-azetidinesulfonic acid and 4-substituted derivatives E.R. Squibb & Sons, Inc. (US) 1983-08-24 EP disclosed
US-4386034-A Sulfamated amino acid amides E. R. SQUIBB & SONS, INC. (US) 1983-05-31 US disclosed
EP-0048953-A2 Beta-lactam antibiotics E.R. Squibb & Sons, Inc. (US) 1982-04-07 EP disclosed