SCHEMBL4524045

SCHEMBL4524045

OCCCCNCc1c(-c2ccccc2)ccnc1Cl

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 2/20 0.40
PDCD1 Q15116 5/20 0.40
CD274 Q9NZQ7 5/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C19 P33261 1/20 0.40
HIF1A Q16665 1/20 0.38
LMNA P02545 1/20 0.38
HDAC3 O15379 1/20 0.38
HDAC4 P56524 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC7 Q8WUI4 1/20 0.38
HDAC2 Q92769 1/20 0.38
HDAC10 Q969S8 1/20 0.38
HDAC11 Q96DB2 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
HDAC9 Q9UKV0 1/20 0.38
HDAC5 Q9UQL6 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4509956 0.96 PDCD1 (0.41) ADORA1PDCD1CD274CYP1A2CYP3A4
SCHEMBL4525266 0.90 CD274 (0.48) PDCD1CD274MEN1KMT2ASMN1; SMN2
SCHEMBL4514401 0.87 CHRM2 (0.38) CYP1A2CYP3A4CYP2D6CYP2C19LMNA
SCHEMBL4516325 0.83 VSIR (0.40) ADORA1PDCD1CD274
SCHEMBL4512711 0.79 PRMT5 (0.41) PDCD1CD274CYP1A2CYP3A4CYP2D6
SCHEMBL4517460 0.77 VSIR (0.45) PDCD1CD274
SCHEMBL4525368 0.77 CD274 (0.36) PDCD1CD274CYP3A4LMNAMEN1
SCHEMBL2511037 0.76 FYN (0.39) CYP1A2CYP2C19LMNAMEN1KMT2A
Hydrochloric Acid SCHEMBL4520463 0.71 LRRK2 (0.38) CYP1A2CYP3A4CYP2D6CYP2C19MEN1
SCHEMBL27319872 0.69 CSNK2A1 (0.54) CD274CYP1A2CYP3A4CYP2D6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7625887-B2 Receptor agonists TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-12-01 US disclosed
US-20060199795-A1 Receptor agonists TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2006-09-07 US disclosed
EP-1591120-A1 RECEPTOR AGONISTS Takeda Chemical Industries, Ltd. (JP) 2005-11-02 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060199795-A1 Receptor agonists GPBAR1, GPR35, GPR55 ADORA1 129/4885PDCD1 4197/4885CD274 3690/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.