SCHEMBL4525591

SCHEMBL4525591

Cc1cccc2cc(C3=NC(C)(C)C(C)c4c(F)cccc43)cnc12

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 5/20 0.35
MGAM O43451 1/20 0.32
GAA P10253 1/20 0.32
SI P14410 1/20 0.32
MGAM2 Q2M2H8 1/20 0.32
ABCB1 P08183 1/20 0.32
ABCG2 Q9UNQ0 1/20 0.32
NPC1 O15118 1/20 0.31
GRIN2B Q13224 2/20 0.31
ATM Q13315 1/20 0.30
PARP1 P09874 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4525440 0.86 HPGDS (0.40)
SCHEMBL4525997 0.84 BRD4 (0.41) NPC1
SCHEMBL20300819 0.81 MGAM (0.33) MGAMGAASIMGAM2NPC1
SCHEMBL4416025 0.79 MGAM (0.36) ABL1MGAMGAASIMGAM2
SCHEMBL29919696 0.79 MGAM (0.36) ABL1MGAMGAASIMGAM2
SCHEMBL31414106 0.78 ABCB1 (0.33) MGAMGAASIMGAM2ABCB1
SCHEMBL20301306 0.77 NPC1 (0.43) NPC1
SCHEMBL31414124 0.77 MGAM (0.35) ABL1MGAMGAASIMGAM2
SCHEMBL4510196 0.77 ALDH1A1 (0.40) ABL1MGAMGAASIMGAM2
SCHEMBL20301317 0.75 NPC1 (0.33) NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7632783-B2 fungicides, pesticides for protecting rice crop, tomatoes, cucumbers and green beans; 3-(5-fluoro-3,3-dimethyl-3,4-dihydroisoquinolin-1-yl)quinoline MITSUI CHEMICALS AGRO, INC. (JP) 2009-12-15 US disclosed
US-20080275242-A1 3-(Dihydro(Tetrahydro)Isoquinolin-1-Yl)Quinoline Compound MITSUI CHEMICALS CROP & LIFE SOLUTIONS, INC. (JP) 2008-11-06 US disclosed
EP-1736471-A1 3-(DIHYDRO(TETRAHYDRO)ISOQUINOLIN-1-YL)QUINOLINES Sankyo Agro Company, Limited (JP) 2006-12-27 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080275242-A1 3-(Dihydro(Tetrahydro)Isoquinolin-1-Yl)Quinoline Compound QTRT1, RABL3, RECQL ABL1 271/4885MGAM 3309/4885GAA 3783/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.