SCHEMBL4528212

SCHEMBL4528212

NC1(CNC(=O)c2cn(-c3ncccn3)c3nccc(Cl)c23)CCCCCC1

nearest known ligand 0.42

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 17/20 0.42
IL1B P01584 5/20 0.40
NTRK1 P04629 1/20 0.38
HCN4 Q9Y3Q4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4535427 0.89 P2RX7 (0.54) P2RX7IL1B
SCHEMBL11026570 0.89 P2RX7 (0.54) P2RX7IL1B
SCHEMBL4540743 0.87 HTR3E (0.43) P2RX7IL1BHCN4
SCHEMBL4364472 0.86 P2RX7 (0.51) P2RX7IL1B
SCHEMBL13706802 0.85 P2RX7 (0.46) P2RX7IL1BHCN4
SCHEMBL4527104 0.85 P2RX7 (0.40) P2RX7IL1BHCN4
SCHEMBL13706906 0.83 HCN4 (0.51) P2RX7HCN4
SCHEMBL4350376 0.83 HCN4 (0.60) P2RX7HCN4
SCHEMBL13706843 0.83 ALDH1A1 (0.56) P2RX7IL1BHCN4
SCHEMBL13706858 0.83 HCN4 (0.60) P2RX7HCN4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009108551-A2 HETEROARYL AMIDE ANALOGUES H. LUNDBECK A/S (DK) 2009-09-03 WO disclosed
WO-2009108551-A2 HETEROARYL AMIDE ANALOGUES H. LUNDBECK A/S (DK) 2009-09-03 WO disclosed