SCHEMBL4530544

SCHEMBL4530544

CCCCCC1=COc2ccccc2C1

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.37
MAOB P27338 1/20 0.37
CYP2D6 P10635 2/20 0.36
ALDH1A1 P00352 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C19 P33261 1/20 0.36
DRD2 P14416 1/20 0.35
SLC6A2 P23975 1/20 0.35
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35
SLC6A4 P31645 1/20 0.35
LIPG Q9Y5X9 1/20 0.33
CYP1A1 P04798 1/20 0.33
KCNH2 Q12809 3/20 0.33
HTT P42858 1/20 0.32
LMNA P02545 1/20 0.32
GAA P10253 1/20 0.32
SIGMAR1 Q99720 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL293444 0.84 MAOA (0.37) MAOAMAOB
SCHEMBL295082 0.83 MAOA (0.36) MAOAMAOB
SCHEMBL511051 0.82 MAOA (0.38) MAOAMAOB
SCHEMBL294572 0.78 MAOA (0.41) MAOAMAOB
SCHEMBL1648706 0.74 KEAP1 (0.43) MAOAMAOBALDH1A1CYP1A2HTT
SCHEMBL295033 0.74 MAOA (0.43) MAOAMAOB
SCHEMBL7977979 0.74 MAOA (0.43) MAOAMAOB
SCHEMBL21615077 0.73 MAOA (0.39) MAOAMAOB
SCHEMBL5613920 0.71 HTR2A (0.48) MAOAMAOBCYP2D6ALDH1A1CYP1A2
SCHEMBL29922564 0.70 HTR2A (0.47) CYP2D6ALDH1A1CYP1A2CYP2C19DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009078029-A2 AN IMPROVED PROCESS FOR THE PREPARATION OF TRANS 3,4- DIARYLCHROMAN AND THEIR DERIVATIVES COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2009-06-25 WO claimed
CN-102850336-A DERIVATIVES OF 4-PIPERAZIN-1-YL-4-BENZ0 [B] THIOPHENE SUITABLE FOR THE TREATMENT OF CNS DISORDERS OTSUKA PHARMA CO LTD 2013-01-02 CN disclosed
CN-102702182-A Derivatives of 4-piperazin-1-yl-4-benzo[b]thiophene suitable for the treatment of cns disorders OTSUKA PHARMA CO LTD 2012-10-03 CN disclosed
CN-102558140-A Derivatives of 4-piperazin-1-1-yl-4-benzo [b] thiophene suitable for the treatment of cns disorders OTSUKA PHARMA CO LTD 2012-07-11 CN disclosed
CN-101258147-B 4-piperazin-1-yl-4-benzo [ B ] thiophene derivatives for the treatment of CNS disorders OTSUKA PHARMA CO LTD 2012-03-21 CN disclosed
WO-2009078029-A2 AN IMPROVED PROCESS FOR THE PREPARATION OF TRANS 3,4- DIARYLCHROMAN AND THEIR DERIVATIVES COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2009-06-25 WO disclosed
CN-101258147-A 4-piperazin-1-yl-4-benzo [ B ] thiophene derivatives for the treatment of CNS disorders OTSUKA PHARMA CO LTD (JP) 2008-09-03 CN disclosed