SCHEMBL4535453

SCHEMBL4535453

O=C(NCC1CCN(S(=O)(=O)c2ccc(-c3ccccc3)cc2)C1)N[C]1CCCCCCC1.[CH2].[CH2]

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.56
L3MBTL1 Q9Y468 1/20 0.56
NAMPT P43490 4/20 0.47
AKR1C3 P42330 1/20 0.47
AKR1C1 Q04828 1/20 0.47
GAA P10253 1/20 0.43
POLB P06746 1/20 0.43
LMNA P02545 2/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
KDM4E B2RXH2 1/20 0.42
TP53 P04637 1/20 0.42
MAPT P10636 1/20 0.42
ALOX15 P16050 1/20 0.42
HTT P42858 1/20 0.42
RECQL P46063 1/20 0.42
EPHX1 P07099 1/20 0.42
MMP2 P08253 1/20 0.42
MMP9 P14780 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4537356 0.94 ALDH1A1 (0.64) ALDH1A1L3MBTL1NAMPTGAAPOLB
SCHEMBL4535924 0.88 ALDH1A1 (0.59) ALDH1A1L3MBTL1NAMPTGAAPOLB
SCHEMBL4537967 0.88 ALDH1A1 (0.50) ALDH1A1L3MBTL1GAAPOLBLMNA
SCHEMBL4539044 0.88 ALDH1A1 (0.50) ALDH1A1L3MBTL1GAAPOLBLMNA
SCHEMBL4537395 0.85 USP30 (0.50) ALDH1A1L3MBTL1NAMPTGAAMEN1
SCHEMBL4535742 0.85 NPC1 (0.52) ALDH1A1L3MBTL1LMNAMEN1KMT2A
SCHEMBL4542202 0.84 KMT2A (0.49) ALDH1A1L3MBTL1NAMPTGAAPOLB
SCHEMBL4540008 0.84 MEN1 (0.50) ALDH1A1L3MBTL1NAMPTGAAPOLB
SCHEMBL4542924 0.84 CYP3A4 (0.59) ALDH1A1L3MBTL1NAMPTGAALMNA
SCHEMBL4540074 0.82 FBP1 (0.50) ALDH1A1L3MBTL1GAAPOLBLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO claimed
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO disclosed