SCHEMBL4536567

SCHEMBL4536567

CNC[CH]c1ccc(O)c(O)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.52
RAB9A P51151 2/20 0.52
PTGS2 P35354 1/20 0.52
LCK P06239 3/20 0.50
ALDH1A1 P00352 3/20 0.46
CYP3A4 P08684 2/20 0.46
RECQL P46063 1/20 0.46
BLM P54132 3/20 0.45
GFER P55789 3/20 0.45
POLB P06746 2/20 0.45
L3MBTL1 Q9Y468 2/20 0.45
ALPL P05186 1/20 0.45
ALPI P09923 1/20 0.45
ALPG P10696 1/20 0.45
CYP1A2 P05177 4/20 0.44
MAPT P10636 3/20 0.44
HIF1A Q16665 3/20 0.44
HSD17B10 Q99714 3/20 0.44
TP53 P04637 2/20 0.44
ALOX15 P16050 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5065668 0.79 ADRB2 (0.47) KDM4ERAB9APTGS2LCKALDH1A1
SCHEMBL11805095 0.79 KDM4E (0.60) KDM4ERAB9APTGS2LCKALDH1A1
SCHEMBL11520449 0.74 LCK (0.47) KDM4ERAB9ALCKALDH1A1CYP3A4
SCHEMBL21049763 0.74 ALDH1A1 (0.63) KDM4ERAB9APTGS2LCKALDH1A1
SCHEMBL28165888 0.72 KDM4E (0.58) KDM4ERAB9APTGS2LCKALDH1A1
SCHEMBL21412902 0.72 LCK (0.45) KDM4ERAB9APTGS2LCKALDH1A1
Protocatechualdehyde SCHEMBL29196221 0.70 KDM4E (0.91) KDM4ERAB9APTGS2LCKALDH1A1
Protocatechualdehyde SCHEMBL28985147 0.70 KDM4E (0.58) KDM4ERAB9APTGS2LCKALDH1A1
Protocatechualdehyde SCHEMBL27648161 0.69 KDM4E (0.79) KDM4ERAB9APTGS2LCKALDH1A1
SCHEMBL17308143 0.69 EGFR (0.69) KDM4ERAB9ALCKALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2637649-A2 COMPOUNDS AND METHODS FOR TREATING PAIN Akron Molecules GmbH (AT) 2013-09-18 EP disclosed
WO-2012062925-A2 COMPOUNDS AND METHODS FOR TREATING PAIN AKRON MOLECULES GMBH (AT) 2012-05-18 WO disclosed