SCHEMBL4537211

SCHEMBL4537211

CC[C@@H](NC(=O)c1ccc(NCc2ccc(C(=O)OC)cc2)c(N)c1)c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KCNK3 O14649 1/20 0.50
TAOK1 Q7L7X3 1/20 0.46
TAOK3 Q9H2K8 1/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
LNPEP Q9UIQ6 3/20 0.45
ERAP2 Q6P179 2/20 0.45
PPARG P37231 6/20 0.44
NPC1 O15118 1/20 0.43
MAPT P10636 1/20 0.43
RAB9A P51151 1/20 0.43
PTGER4 P35408 2/20 0.42
TAS1R3 Q7RTX0 2/20 0.42
TAS1R1 Q7RTX1 2/20 0.42
ERAP1 Q9NZ08 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4537762 0.92 PPARG (0.48) LNPEPPPARGMAPTHDAC1HDAC8
SCHEMBL8034344 0.89 PPARG (0.54) PPARGMAPTHDAC1
SCHEMBL8032490 0.87 PPARG (0.55) PPARGHDAC1
SCHEMBL8034539 0.85 PPARG (0.56) PPARGTAS1R3TAS1R1HDAC1HDAC8
SCHEMBL4540765 0.85 MEN1 (0.52) PPARGMAPTHDAC1HDAC8HDAC6
SCHEMBL4536613 0.85 MAPT (0.55) KCNK3MAPTRAB9APTGER4
SCHEMBL8028550 0.83 PPARG (0.58) PPARGMAPTTAS1R3TAS1R1
SCHEMBL8040416 0.83 PPARG (0.58) PPARGTAS1R3TAS1R1
SCHEMBL8038740 0.82 PPARG (0.57) PPARG
SCHEMBL8034326 0.82 PPARG (0.48) PPARGTAS1R3TAS1R1HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009083526-A1 NOVEL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2009-07-09 WO disclosed
WO-2009083526-A1 NOVEL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2009-07-09 WO disclosed