SCHEMBL4540765

SCHEMBL4540765

CC[C@@H](NC(=O)c1ccc(NCc2ccc(F)c(F)c2)c(N)c1)c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
PKM P14618 1/20 0.52
PPARG P37231 13/20 0.47
MAPT P10636 2/20 0.47
LMNA P02545 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
HDAC1 Q13547 3/20 0.43
HDAC3 O15379 2/20 0.43
HDAC2 Q92769 2/20 0.43
NCOR2 Q9Y618 2/20 0.43
HDAC8 Q9BY41 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
SLC6A9 P48067 1/20 0.43
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8040416 0.92 PPARG (0.58) MEN1KMT2APKMPPARG
SCHEMBL8034344 0.90 PPARG (0.54) MEN1KMT2APPARGMAPTHDAC1
SCHEMBL4537762 0.89 PPARG (0.48) PPARGMAPTLMNAHDAC1HDAC8
SCHEMBL8034539 0.86 PPARG (0.56) PPARGHDAC1HDAC8HDAC6
SCHEMBL4538730 0.86 PPARG (0.57) PPARGMAPTSMN1; SMN2HDAC1HDAC3
SCHEMBL4537211 0.85 KCNK3 (0.50) PPARGMAPTHDAC1HDAC8HDAC6
SCHEMBL4534800 0.85 KMT2A (0.67) MEN1KMT2APKMMAPT
SCHEMBL8032490 0.84 PPARG (0.55) PPARGHDAC1HDAC3
SCHEMBL8038553 0.84 PPARG (0.60) PPARGHDAC1HDAC3HDAC2NCOR2
SCHEMBL8038556 0.83 PPARG (0.61) PPARGHDAC1HDAC3HDAC2NCOR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009083526-A1 NOVEL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2009-07-09 WO disclosed
WO-2009083526-A1 NOVEL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2009-07-09 WO disclosed