SCHEMBL4537585

SCHEMBL4537585

CC(C)OC(=O)CCC(N)C(=O)OC(C)C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.46
SLC1A1 P43005 2/20 0.36
TSHR P16473 2/20 0.35
MAPT P10636 2/20 0.35
GABRP O00591 2/20 0.34
GABRD O14764 2/20 0.34
GABRA1 P14867 2/20 0.34
GABRB1 P18505 2/20 0.34
GABRG2 P18507 2/20 0.34
GABRB3 P28472 2/20 0.34
GABRA5 P31644 2/20 0.34
GABRA3 P34903 2/20 0.34
GABRA2 P47869 2/20 0.34
GABRB2 P47870 2/20 0.34
GABRA4 P48169 2/20 0.34
GABRE P78334 2/20 0.34
GABRA6 Q16445 2/20 0.34
GABRG1 Q8N1C3 2/20 0.34
GABRG3 Q99928 2/20 0.34
GABRQ Q9UN88 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28096046 1.00 LMNA (0.46) LMNASLC1A1TSHRMAPTGABRP
SCHEMBL2241803 1.00 LMNA (0.46) LMNASLC1A1TSHRMAPTGABRP
SCHEMBL22639581 0.89 SLC1A1 (0.49) LMNASLC1A1TSHRMAPTGABRP
SCHEMBL16523558 0.89 LMNA (0.43) LMNASLC1A1TSHRMAPTGABRP
SCHEMBL16523559 0.87 LMNA (0.46) LMNASLC1A1TSHRGABRPGABRD
SCHEMBL31229067 0.87 CYP1A2 (0.44) LMNASLC1A1GABRPGABRDGABRA1
SCHEMBL14175423 0.87 CYP1A2 (0.44) LMNASLC1A1GABRPGABRDGABRA1
SCHEMBL2201201 0.84 SLC1A1 (0.54) LMNASLC1A1GRM8GRM6GRIN2D
SCHEMBL23515280 0.84 SLC1A1 (0.36) LMNASLC1A1GABRPGABRDGABRA1
SCHEMBL5885314 0.84 SLC1A1 (0.36) LMNASLC1A1GABRPGABRDGABRA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 29 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102796097-B Phenanthroindolizididerivative pyridine alcaloid-derivatives, its preparation method and pharmaceutical composition and purposes INSTITUTE OF MATARIA MEDICA, CHINESE ACADEMY OF MEDICAL SCIENCES (CN) 2016-12-14 CN claimed
EP-1603549-A2 IMPROVED BIOAVAILABILITY AND IMPROVED DELIVERY OF ACIDIC PHARMACEUTICAL DRUGS Yu, Ruey J., Dr. (US) 2005-12-14 EP claimed
US-20040220264-A1 Bioavailability and improved delivery of acidic pharmaceutical drugs YU RUEY J 2004-11-04 US claimed
WO-2004082628-A2 IMPROVED BIOAVAILABILITY AND IMPROVED DELIVERY OF ACIDIC PHARMACEUTICAL DRUGS YU RUEY J (US) 2004-09-30 WO claimed
JP-9143497-A None JP disclosed
CN-108794372-B Novel compound and pharmaceutical composition for treating tuberculosis comprising same 顺天乡大学校产学协力团 2021-09-14 CN disclosed
US-20190292171-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF CANCER CELLIX BIO PRIVATE LIMITED (IN) 2019-09-26 US disclosed
CN-105924380-B Luxuriant and rich with fragrance class compound or derivatives thereof and treatment medicine for tuberculosis compositions containing the phenanthrene class compound or derivatives thereof 顺天乡大学校产学协力团 2019-03-05 CN disclosed
CN-108794372-A New compound and tuberculotherapy medical composition comprising it 顺天乡大学校产学协力团 2018-11-13 CN disclosed
CN-102796097-B Phenanthroindolizididerivative pyridine alcaloid-derivatives, its preparation method and pharmaceutical composition and purposes INSTITUTE OF MATARIA MEDICA, CHINESE ACADEMY OF MEDICAL SCIENCES (CN) 2016-12-14 CN disclosed
CN-101365415-B Gelling agent AJINOMOTO KK 2012-09-12 CN disclosed
US-8084499-B2 Modified clay mineral AJINOMOTO CO., INC. (JP) 2011-12-27 US disclosed
US-4866093-A INHIBITING CHOLESTEROL BIOSYNTHESIS IN THE LIVER SANKYO COMPANY LIMITED (JP) 1989-09-12 US disclosed
US-4695587-A CHOLESTEROL BIOSYNTHESIS INHIBITORS SANKYO COMPANY LIMITED (JP) 1987-09-22 US disclosed
EP-0065835-B1 M-4 AND ISO M-4 DERIVATIVES, THEIR PREPARATION AND COMPOSITIONS CONTAINING THEM SANKYO COMPANY LIMITED (JP) 1985-11-13 EP disclosed
EP-0065843-B1 NEW M-4 AND ISO M-4 DERIVATIVES, THEIR PREPARATION AND COMPOSITIONS CONTAINING THEM SANKYO COMPANY LIMITED (JP) 1985-09-18 EP disclosed
US-4479965-A ANTILIPEMIC, ANTICHOLESTEROL AGENTS SANKYO COMPANY, LIMITED (JP) 1984-10-30 US disclosed
US-4451481-A ANTICHOLESTEROL AGENTS SANKYO COMPANY LIMITED (JP) 1984-05-29 US disclosed
EP-0065835-A1 M-4 and iso M-4 derivatives, their preparation and compositions containing them SANKYO COMPANY LIMITED (JP) 1982-12-01 EP disclosed
EP-0065843-A1 New M-4 and iso M-4 derivatives, their preparation and compositions containing them SANKYO COMPANY LIMITED (JP) 1982-12-01 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190292171-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF CANCER SI, HBG2, HBG1 LMNA 1933/4885SLC1A1 3154/4885TSHR 3208/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.