Acridine

Acridine

SCHEMBL453862

c1c[nH]cn1.c1ccc2nc3ccccc3cc2c1

nearest known ligand 0.58

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.58
HPGD P15428 3/20 0.58
MAPT P10636 3/20 0.58
GLA P06280 2/20 0.58
ACHE P22303 1/20 0.58
FKBP5 Q13451 1/20 0.50
HTR3A P46098 1/20 0.44
NQO2 P16083 1/20 0.40
GAA P10253 3/20 0.39
KMT2A Q03164 3/20 0.39
KDM4E B2RXH2 2/20 0.39
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
LMNA P02545 1/20 0.39
POLB P06746 1/20 0.39
PTBP1 P26599 1/20 0.39
RCE1 Q9Y256 1/20 0.39
PDGFRB P09619 1/20 0.37
PDGFRA P16234 1/20 0.37
PDE2A O00408 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Acridine SCHEMBL29354628 1.00 ALDH1A1 (0.58) ALDH1A1HPGDMAPTGLAACHE
Acridine SCHEMBL28281831 0.98 ALDH1A1 (0.56) ALDH1A1HPGDMAPTGLAACHE
Phenazine SCHEMBL28557583 0.88 ALDH1A1 (0.59) ALDH1A1HPGDMAPTGLAACHE
Anthracene SCHEMBL28457231 0.88 ALDH1A1 (0.59) ALDH1A1HPGDMAPTGLAACHE
Anthracene SCHEMBL28211461 0.88 ALDH1A1 (0.59) ALDH1A1HPGDMAPTGLAACHE
Acridine SCHEMBL27413186 0.87 CYP1A2 (0.56) ALDH1A1HPGDMAPTGLAACHE
Naphthalene SCHEMBL2123892 0.83 ALDH1A1 (0.65) ALDH1A1FKBP5CYP2A6
Naphthalene SCHEMBL338629 0.83 ALDH1A1 (0.65) ALDH1A1FKBP5CYP2A6
Naphthalene SCHEMBL27481708 0.81 ALDH1A1 (0.62) ALDH1A1FKBP5CYP2A6
Cinnoline SCHEMBL10732584 0.80 ALDH1A1 (0.45) ALDH1A1HPGDMAPTGLAACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 75 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109069470-A Use of specific benzodihydrofuran lignans for inhibiting breast cancer cell metastasis 杨宁荪 2018-12-21 CN claimed
CN-108440565-A A kind of luxuriant receptor of acridine imidazoles ring of naphthalene nucleus bridging and preparation method thereof and the identification application to iron ion and dihydrogen phosphate ions 福州大学 2018-08-24 CN claimed
WO-2023202686-A1 COMPOSITION AND METHOD FOR INHIBITING XANTHINE DEHYDROGENASE (XDH) 上海舶望制药有限公司 2023-10-26 WO disclosed
CN-114525280-A iRNA compositions of programmed cell death 1 ligand 1(PD-L1) and methods of use thereof 阿尔尼拉姆医药品有限公司 2022-05-24 CN disclosed
CN-108368507-B iRNA compositions of programmed cell death 1 ligand 1(PD-L1) and methods of use thereof 阿尔尼拉姆医药品有限公司 2022-03-22 CN disclosed
CN-110461876-A For exhausting the composition and method of CD137+ cell MAGENTA THERAPEUTICS INC 2019-11-15 CN disclosed
CN-109661400-A Compositions and methods for depleting CD117+ cells 美真达治疗公司 2019-04-19 CN disclosed
CN-109641051-A For exhausting the composition and method of cell 美真达治疗公司 2019-04-16 CN disclosed
CN-109462995-A The method and composition of bioactivator 波涛生命科学有限公司 2019-03-12 CN disclosed
CN-109069470-A Use of specific benzodihydrofuran lignans for inhibiting breast cancer cell metastasis 杨宁荪 2018-12-21 CN disclosed
CN-108602849-A For by RNA nanotechnologies by the RNA ligand presen-tation allochthons of therapeutic agent specific delivery to cell 俄亥俄州国家创新基金会 2018-09-28 CN disclosed
CN-1701063-A Therapeutic acridone and acridine compounds CANCER REC TECH LTD (GB) 2005-11-23 CN disclosed
CN-1652772-A (+) -2- [ 1- (3-ethoxy-4-methoxyphenyl) -2-methylsulfonylethyl ] -4-acetylaminoisoindoline-1, 3-dione, methods of use, and compositions thereof CELGENE CORP (US) 2005-08-10 CN disclosed
US-20050070568-A1 Therapeutic acridone and acridine compounds CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2005-03-31 US disclosed
CN-1568188-A Nociceptin analogs EURO CELTIQUE SA (LU) 2005-01-19 CN disclosed
CN-1561211-A Nociceptin analogs EURO CELTIQUE SA (LU) 2005-01-05 CN disclosed
EP-1474397-A1 THERAPEUTIC ACRIDONE AND ACRIDINE COMPOUNDS Cancer Research Technology Limited (GB) 2004-11-10 EP disclosed
CN-1516584-A Spiropyrazole compounds ŷ�����ǹɷ����޹�˾ 2004-07-28 CN disclosed
WO-2003059885-A1 THERAPEUTIC ACRIDONE AND ACRIDINE COMPOUNDS CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2003-07-24 WO disclosed
WO-2002079380-A2 DISRUPTIONS IN GABA RECEPTOR RH02 SUBUNIT, METHODS ADN USES THEREOF DELTAGEN, INC. (US) 2002-10-10 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050070568-A1 Therapeutic acridone and acridine compounds CCNK, TERT, CCNA1 ALDH1A1 99/4885HPGD 709/4885MAPT 3941/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.