SCHEMBL4539282

SCHEMBL4539282

N=C(N)C1=COc2ccccc2C1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 2/20 0.41
MAOB P27338 1/20 0.41
NISCH Q9Y2I1 2/20 0.40
F2 P00734 1/20 0.33
F10 P00742 1/20 0.33
F12 P00748 1/20 0.33
F7 P08709 1/20 0.33
F3 P13726 1/20 0.33
PKM P14618 1/20 0.33
BLM P54132 1/20 0.32
TMPRSS2 O15393 1/20 0.32
HTR1A P08908 1/20 0.32
ADRA2A P08913 1/20 0.32
CYP2D6 P10635 1/20 0.32
SLC6A2 P23975 1/20 0.32
OXTR P30559 1/20 0.32
PRSS1 P07477 1/20 0.31
PRSS2 P07478 1/20 0.31
C1S P09871 1/20 0.31
PRSS3 P35030 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2230058 0.82 MAOA (0.41) MAOAMAOBNISCHBLMOXTR
SCHEMBL212723 0.76 MAOA (0.42) MAOAMAOBOXTR
SCHEMBL16397646 0.76 MAOA (0.42) MAOAMAOBOXTR
SCHEMBL9058873 0.75 MAOA (0.41) MAOAMAOBOXTR
Trifluoroacetic Acid SCHEMBL16669664 0.73 MAOA (0.33) MAOAMAOBF2BLMPRSS1
SCHEMBL18280613 0.71 MAOA (0.48) MAOAMAOBNISCHCYP2D6OXTR
SCHEMBL30714851 0.71 MAOA (0.48) MAOAMAOBNISCHOXTR
SCHEMBL1707855 0.71 MAOA (0.48) MAOAMAOBNISCHOXTR
SCHEMBL2013569 0.71 MAOA (0.48) MAOAMAOBNISCHOXTR
SCHEMBL295062 0.69 MAOA (0.50) MAOAMAOBOXTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2638025-A2 CHROMENE DERIVATIVES AND THEIR ANALOGA AS WNT PATHWAY ANTAGONISTS Deutsches Krebsforschungszentrum (DKFZ) (DE) 2013-09-18 EP disclosed
WO-2012062901-A2 CHROMENE DERIVATIVES AND THEIR ANALOGA AS WNT PATHWAY ANTAGONISTS DEUTSCHES KREBSFORSCHUNGSZENTRUM (DKFZ) (DE) 2012-05-18 WO disclosed